| Identification | Back Directory | [Name]
3-[4-(Hexyloxy)-1,2,5-thiadiazol-3-yl]-1,2,5,6-tetrahydro-1-methylpyridineoxalate | [CAS]
141064-23-5 | [Synonyms]
Lumeron
LY246708 oxalate
Xanomeline oxalate
Xanomeline oxalate salt
LY246708;MEMCOR;LUMERON
3-(3-Hexyloxy-1,2,5-thiadiazol-4-yl)-1,2,5,6-tetrahydro-1-methylpyridine oxalate
3-[4-(Hexyloxy)-1,2,5-thiadiazol-3-yl]-1,2,5,6-tetrahydro-1-methylpyridineoxalate
3-[4-(Hexyloxy)-1,2,5-thiadiazol-3-yl]-1,2,5,6-tetrahydro-1-methylpyridine ethanedioate (1:1) | [Molecular Formula]
C14H23N3OS.C2H2O4 | [MDL Number]
MFCD12828778 | [MOL File]
141064-23-5.mol | [Molecular Weight]
371 |
| Chemical Properties | Back Directory | [Melting point ]
148-150℃ | [storage temp. ]
Desiccate at +4°C | [solubility ]
DMF: 1.6 mg/ml; DMF:PBS (pH 7.2) (1:9): 0.1 mg/ml | [form ]
Powder |
| Hazard Information | Back Directory | [Description]
Muscarinic receptors are G protein-coupled acetylcholine receptors that play diverse roles. Xanomeline (oxalate) is a potent agonist of muscarinic acetylcholine receptors (EC50 values are 0.3, 92.5, 5, 52, and 42 nM for M1, M2, M3, M4, and M5, respectively). It has antipsychotic-like activities in rats and Cebus monkeys. M1 selective agonists, like Xanomeline (oxalate), enhance memory function and has utility in treating Alzheimer’s Disease. | [Uses]
Xanomeline oxalate is a functionally selective mAChR M1 agonist. | [storage]
Store at -20°C |
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| Company Name: |
SPIRO PHARMA
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| Tel: |
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| Website: |
www.spiropharma.com.cn |
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