ADRA1D receptor agonist 1
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- CAS号:
- 1191908-14-1
- 英文名:
- ADRA1D receptor agonist 1
- 英文别名:
- ADRA1D receptor agonist 1;ADRA1D receptor antagonist 1;ADRA1D receptor antagonist 1 HCl;ADRA-1D receptor antagonist 1,ADRA1D receptor antagonist 1
- 中文名:
- ADRA1D receptor agonist 1
- 中文别名:
- 化合物 T10250;ADRA1D RECEPTOR ANTAGONIST 1 盐酸盐
- CBNumber:
- CB78054299
- 分子式:
- C15H14Cl2N4O
- 分子量:
- 337.2
- MOL File:
- 1191908-14-1.mol
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ADRA1D receptor agonist 1化学性质
ADRA1D receptor agonist 1性质、用途与生产工艺
ADRA1D receptor agonist 1 (compound (R)-9S) 是一个高效、选择性的，有口服活性的 α1D 肾上腺素受拮抗剂，Ki 值为 1.6 nM。
Ki: 1.6 nM (α
1D
adrenoceptor)
ADRA1D receptor agonist 1 shows low hERG inhibition.
ADRA1D receptor agonist 1 exhibits higher selectivity for α1D-AR over α1A- and α1B-ARs .
ADRA1D receptor agonist 1 (4.4 µg/kg; i.v.) dose-dependently decreases the non-voiding bladder contractions during the urinary storage phase in rats with BOO.
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Animal Model:
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Rat with bladder outlet obstruction (BOO)
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Dosage:
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4.4 µg/kg
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Administration:
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Intravenous injection
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Result:
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Dose-dependently decreased the non-voiding bladder contractions during urinary storage phase in rats with BOO.
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ADRA1D receptor agonist 1
上下游产品信息
上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
|---|
| 2024/04/30 | HY-135270 | ADRA1D receptor antagonist 1 | | 1 mg | 2181元 |
| 2024/04/30 | HY-135270 | ADRA1D receptor antagonist 1 | | 5 mg | 4800元 |
ADRA1D receptor agonist 1
生产厂家
1191908-14-1, ADRA1D receptor agonist 1 相关搜索:
- ADRA1D RECEPTOR ANTAGONIST 1 盐酸盐
- 化合物 T10250
- 1191908-14-1
- ADRA1D receptor antagonist 1 HCl
- ADRA-1D receptor antagonist 1,ADRA1D receptor antagonist 1
- ADRA1D receptor antagonist 1
- ADRA1D receptor agonist 1