857876-30-3 Basic information More..
Product Name:AMG-706
Synonyms:Motesanib, Diphosphate Salt;AMG-706;Motesanib(AMG-706);Motesanib diphosphate;Motesanib diphosphate [usan];Unii-T6Q3060U91;N-(2,3-Dihydro-3,3-dimethyl-1H-indol-6-yl)-2-[(4-pyridinylmethyl)amino]-3-pyridinecarboxamide diphosphate;N-(2,3-Dihydro-3,3-diMethyl-1H-indol-6-yl)-2-[(4-pyridinylMethyl)aMino]-3-pyridinecarboxaMide Phosphate
CAS:857876-30-3
MF:C22H29N5O9P2
MW:569.441282
EINECS:
Mol File:857876-30-3.mol
857876-30-3

Use

Motesanib Diphosphate (AMG-706) is a potent ATP-competitive inhibitor of VEGFR1/2/3, PDGFR, c-Kit and Ret with IC50 of 2 nM/3 nM/6 nM, 84 nM, 8 nM and 59 nM, respectively.

AMG-706 manufacturers

  • AMG-706
  • US $2.00 / kg
  • 2019-07-06
  • CAS:857876-30-3
  • Min. Order: 1kg
  • Purity: 99%
  • Supply Ability: 100kg
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