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| Product Name: | ARN272 | | Synonyms: | CS-2535;4-[[4-(4-Hydroxyphenyl)-1-phthalazinyl]amino]-N-phenylbenzamide;Benzamide, 4-[[4-(4-hydroxyphenyl)-1-phthalazinyl]amino]-N-phenyl-;4-(4-(4-hydroxyphenyl)phthalazin-1-ylamino)-N-phenylbenzamide;ARN272,inhibit,Inhibitor,ARN-272 | | CAS: | 488793-85-7 | | MF: | C27H20N4O2 | | MW: | 432.47 | | EINECS: | | | Product Categories: | | | Mol File: | 488793-85-7.mol |  |
| | ARN272 Chemical Properties |
| storage temp. | Store at -20°C | | solubility | Soluble in DMSO |
| | ARN272 Usage And Synthesis |
| Description | ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor. ARN272 attenuates nausea-induced behaviour in rats, and vomiting in shrews (Suncus murinus). The anandamide transport inhibition by ARN272 tonically activates CB1 receptors and as such produces a type of indirect agonism to regulate toxin-induced nausea and vomiting. |
| | ARN272 Preparation Products And Raw materials |
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