| Identification | Back Directory | [Name]
THIETHYLPERAZINE MALEATE (200 MG) | [CAS]
1179-69-7 | [Synonyms]
gs-95
torecan
tresten
toresten
nsc-130044
torecanmaleate
2-butenedioate
torecanbimaleate
torecandimaleate
(z)-10h-phenothiazin
thiethylperazinemaleate
thiethylperazinedimaleate
THIETHYLPERAZINE MALEATE (200 MG)
thiethylperazine di(hydrogen maleate)
2-(ethylthio)-10-(3-(4-methyl-1-piperazinyl)propyl)-phenothiazindimaleat
2-(ethylthio)-10-(3-(4-methyl-1-piperazinyl)propyl)phenothiazinedimaleate
2-(ethylthio)-10-(3-(4-methyl-1-piperazinyl)propyl)-phenothiazinmaleate(1
3-ethylmercapto-10-(1’-methylpiperazinyl-4’-propyl)phenothiazinedimaleate
2-ethylmercapto-10-(3-(1-methyl-4-piperazinyl)propyl)phenothiazinedimaleate
2-(ethylthio)-10-(3-(4-methyl-1-piperazinyl)propyl)phenothiazinemaleate(1:2
2-(ethylthio)-10-(3-(4-methyl-1-piperazinyl)propyl)-phenothiazinmaleate(1:2) | [EINECS(EC#)]
214-648-9 | [Molecular Formula]
C4H2O4-2 | [MDL Number]
MFCD01706868 | [MOL File]
1179-69-7.mol | [Molecular Weight]
114.056 |
| Chemical Properties | Back Directory | [Melting point ]
>146oC (dec.) | [storage temp. ]
Hygroscopic, -20°C Freezer, Under inert atmosphere | [solubility ]
DMSO (Slightly), Methanol (Slightly, Heated) | [form ]
Solid | [color ]
Off-White to Pale Yellow | [Stability:]
Hygroscopic |
| Hazard Information | Back Directory | [Uses]
Thiethylperazine Maleate is used a phenothiazine derivative used in the treatment of multi-drug resistant (MDR) bacterial infections. Antibacterial. | [in vivo]
Thiethylperazine (3 mg/kg; intramuscular injection; twice daily; for 30 days; young APP/PS1 mice) treatment significantly reduces Aβ42 levels in APP/PS1 mice[2]. | Animal Model: | Young Aβ precursor protein (APPswe) and mutant presenilin-1 (PS1) (APP/PS1) mice[2] | | Dosage: | 3 mg/kg | | Administration: | Intramuscular injection; twice daily; for 30 days | | Result: | Significantly reduced Aβ42 levels in APP/PS1 mice.
|
| [IC 50]
D2 Receptor; H1 Receptor | [storage]
4°C, away from moisture and light |
|
| Company Name: |
Wuhan Topule
|
| Tel: |
+86-02787215551 19945035818 |
| Website: |
www.topule.com/ |
| Company Name: |
cjbscvictory
|
| Tel: |
13348960310 13348960310; |
| Website: |
https://www.weikeqi-biotech.com/ |
|