| Identification | Back Directory | [Name]
5-HYDROXYMETHYL TOLTERODINE-D14 | [CAS]
1191280-58-6 | [Synonyms]
5-HYDROXYMETHYL TOLTERODINE-D14
Tolterodine 5-Hydroxymethyl-d14 (racemate, as HCl salt)
[2H14]-Tolterodine 5-Hydroxymethyl (racemate, as HCl salt) | [Molecular Formula]
C22H31NO2 | [MOL File]
1191280-58-6.mol | [Molecular Weight]
341.5 |
| Hazard Information | Back Directory | [Uses]
5-HYDROXYMETHYL TOLTERODINE-D14 is intended for use as an internal standard for the quantification of Tolterodine by GC- or LC-mass spectrometry.
| [in vivo]
Desfesoterodine (PNU-200577; 5-Hydroxymethyl Tolterodine; 0.1 and 1 mg/kg; IV) significantly increases bladder compliance after moderate and high doses[5].
In vivo, Desfesoterodine is significantly more potent at suppressing acetylcholine-induced urinary bladder contraction than electrically induced salivation in the anaesthetised cat (ID50=15 and 40 nmol/kg, respectively) [2].
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