| Identification | Back Directory | [Name]
2H-1-Benzopyran-2-one, 7-(1,1-dimethyloctyl)-5-hydroxy-3-[(2-hydroxyphenyl)methyl]- | [CAS]
1399049-81-0 | [Synonyms]
PSB-SB-487
5-hydroxy-3-(2-hydroxybenzyl)-7-(2-methylnonan-2-yl)-2H-chromen-2-one
2H-1-Benzopyran-2-one, 7-(1,1-dimethyloctyl)-5-hydroxy-3-[(2-hydroxyphenyl)methyl]- | [Molecular Formula]
C26H32O4 | [MOL File]
1399049-81-0.mol | [Molecular Weight]
408.53 |
| Chemical Properties | Back Directory | [Boiling point ]
580.4±50.0 °C(Predicted) | [density ]
1.147±0.06 g/cm3(Predicted) | [form ]
Solid | [pka]
7.53±0.20(Predicted) | [color ]
White to off-white |
| Hazard Information | Back Directory | [Uses]
PSB-SB-487 is a potent GPR55 antagonist and CB2 agonist with an IC50 value of 0.113 μM for GPR55, and a Ki value of 0.292 μM for human CB2. PSB-SB-487 can be used for researching diabetes, Parkinson’s disease, neuropathic pain, and cancer[1]. | [References]
[1] Viktor Rempel, et al. Antagonists for the orphan G-protein-coupled receptor GPR55 based on a coumarin scaffold. J Med Chem. 2013 Jun 13;56(11):4798-810. DOI:10.1021/jm4005175 |
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| Company Name: |
cjbscvictory
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| Telephone: |
13348960310 13348960310 |
| Website: |
www.weikeqi-biotech.com/ |
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