| Identification | Back Directory | [Name]
(3-HYDROXYPHENYL)-1,2,3,4,4A,5,12,12AA-OCTAHYDROQUINOLINO[2,3,3-G]ISOQUINOLINE DIHYDROBROMIDE | [CAS]
148545-09-9 | [Synonyms]
SB-205607
TAN-67 HYDROBROMIDE
SB 205607 dihydrobro
TAN-67 DIHYDROBROMIDE
SB 205607 DIHYDROBROMIDE
(3-HYDROXYPHENYL)-1,2,3,4,4A,5,12,12AA-OCTAHYDROQUINOLINO[2,3,3-G]ISOQUINOLINE DIHYDROBROMIDE
Phenol, 3-[(4aR,12aS)-1,3,4,5,12,12a-hexahydro-2-methylpyrido[3,4-b]acridin-4a(2H)-yl]-, rel-
2-Methyl-4aa-(3-hydroxyphenyl)-1,2,3,4,4a,5,12,12aa-octahydroquinolino[2.3.3-g]isoquinolinedihydrobromide]
2-METHYL-4AA-(3-HYDROXYPHENYL)-1,2,3,4,4A,5,12,12AA-OCTAHYDROQUINOLINO[2,3,3-G]ISOQUINOLINE DIHYDROBROMIDE
(R*,S*)-(±)-2-Methyl-4aa-(3-hydroxyphenyl)-1,2,3,4,4a,5,12,12aa-octahydroquinolino[2,3,3-g]isoquinolinedihydrobromide
SB-205607 dihydrobromide, (3-Hydroxyphenyl)-1,2,3,4,4a,5,12,12aa-octahydroquinolino[2,3,3-g]isoquinoline dihydrobromide | [Molecular Formula]
C23H24N2O | [MDL Number]
MFCD05865267 | [MOL File]
148545-09-9.mol | [Molecular Weight]
344.45 |
| Chemical Properties | Back Directory | [Boiling point ]
528.2±50.0 °C(Predicted) | [density ]
1.212±0.06 g/cm3(Predicted) | [storage temp. ]
2-8°C | [solubility ]
H2O: ~15 mg/mL, soluble | [form ]
solid | [pka]
9.92±0.10(Predicted) | [color ]
off-white |
| Hazard Information | Back Directory | [Uses]
SB 205607 Dihydrobromide is a selective δ-opioid receptor-1 agonist. | [Biological Activity]
The first described non-peptide δ 1 opioid receptor agonist with very high affinity and selectivity for the δ 1 subtype (K i values are 1.12, 2320 and 1790 nM at δ 1 , μ and κ receptors respectively). |
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