| Identification | Back Directory | [Name]
U 93631 | [CAS]
152273-12-6 | [Synonyms]
U 93631
CS-2235
U-93631; U 93631
tert-butyl 4,4-dimethyl-5H-imidazo[1,5-a]quinoxaline-3-carboxylate
4,5-Dihydro-4,4-dimethyl-imidazo[1,5-a]quinoxaline-3-carboxylicacid1,1-dimethylethylester
Imidazo(1,5-a)quinoxaline-3-carboxylic acid, 4,5-dihydro-4,4-dimethyl-, 1,1-dimethylethyl ester | [Molecular Formula]
C17H21N3O2 | [MDL Number]
MFCD10566712 | [MOL File]
152273-12-6.mol | [Molecular Weight]
299.37 |
| Chemical Properties | Back Directory | [storage temp. ]
Keep in dark place,Inert atmosphere,2-8°C | [solubility ]
DMF: 25 mg/ml; DMSO: 20 mg/ml; Ethanol: 20 mg/ml | [form ]
A crystalline solid | [color ]
White to off-white |
| Hazard Information | Back Directory | [Uses]
U 93631 is a GABAA receptor antagonist picrotoxin, which inhibits 5-hydroxytryptamine type 3A receptors. | [Biological Activity]
GABA A receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction. Accelerates the decay of GABA-induced Cl - currents with little effect on peak amplitude. Also inhibits 5-HT 3A receptors via a similar mechanism. |
|
|