| Identification | Back Directory | [Name]
Cyclohexanecarboxamide, N-[5-(3,4-dimethoxyphenyl)thieno[2,3-b]pyridin-3-yl]- | [CAS]
1629227-34-4 | [Synonyms]
DRAK1/2-IN-1
Dual DRAK1 and DRAK2 inhibitor 1
Cyclohexanecarboxamide, N-[5-(3,4-dimethoxyphenyl)thieno[2,3-b]pyridin-3-yl]- | [Molecular Formula]
C22H24N2O3S | [MOL File]
1629227-34-4.mol | [Molecular Weight]
396.5 |
| Hazard Information | Back Directory | [Uses]
DRAK1/2-IN-1 (compound 10e) is an active dual DRAK1 and DRAK2 inhibitor with Kd values of 1 μM and 6 μM, respectively[1]. | [References]
[1] Gao LJ, et al. Discovery of dual death-associated protein related apoptosis inducing protein kinase 1 and 2 inhibitors by a scaffold hopping approach. J Med Chem. 2014 Sep 25;57(18):7624-43. DOI:10.1021/jm5007929 |
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