| Identification | Back Directory | [Name]
L-759,656 | [CAS]
174627-56-6 | [Synonyms]
656
L-759,656
(6aR,10aR)-3-(1,1-Dimethylheptyl)-6a,7,8,9,10,10a-hexahydro-1-methoxy-6,6-dimethyl-9-methylene-6H-dibenzo[b,d]pyran | [Molecular Formula]
C26H40O2 | [MDL Number]
MFCD05662267 | [MOL File]
174627-56-6.mol | [Molecular Weight]
384.59 |
| Hazard Information | Back Directory | [Uses]
L-759,656 is a potent CB2-selective annabinoid receptor antagnoist. | [Biological Activity]
Highly selective CB 2 receptor agonist (K i values are 11.8 and 4888 nM for CB 2 and CB 1 receptors respectively). Potently inhibits forskolin-stimulated cAMP production via CB 2 receptors expressed in CHO cells (EC 50 = 3.1 nM). |
|
|