| Chemical Properties | Back Directory | [Boiling point ]
889.930±65.00 °C(Press: 760.00 Torr)(predicted) | [density ]
1.175±0.06 g/cm3(Temp: 25 °C; Press: 760 Torr)(predicted) | [form ]
Solid | [pka]
12.947±0.46(predicted) | [color ]
White to off-white |
| Hazard Information | Back Directory | [Uses]
LU-002i is a subunit-selective human proteasome β2c and β2i inhibitor with an IC50 value of 220 nM for β2i[1]. | [References]
[1] Xin BT, et al. Structure-Based Design of Inhibitors Selective for Human Proteasome β2c or β2i Subunits. J Med Chem. 2019 Feb 14;62(3):1626-1642. DOI:10.1021/acs.jmedchem.8b01884 |
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