| Identification | Back Directory | [Name]
3,5-Pyridinedicarboxylic acid, 1,4-dihydro-2-methyl-6-phenyl-4-[(1E)-2-phenylethenyl]-, 3,5-diethyl ester | [CAS]
185259-16-9 | [Synonyms]
MRS1097
MRS-1097
MRS 1097
3,5-Pyridinedicarboxylic acid, 1,4-dihydro-2-methyl-6-phenyl-4-[(1E)-2-phenylethenyl]-, 3,5-diethyl ester | [Molecular Formula]
C26H27NO4 | [MOL File]
185259-16-9.mol | [Molecular Weight]
417.5 |
| Chemical Properties | Back Directory | [Melting point ]
123-124 °C(Solv: ethyl acetate (141-78-6); hexane (110-54-3)) | [Boiling point ]
566.6±50.0 °C(Predicted) | [density ]
1.187±0.06 g/cm3(Predicted) | [pka]
2.42±0.70(Predicted) |
| Hazard Information | Back Directory | [Description]
MRS1097 is a novel A3 adenosine receptor-selective antagonist. | [Uses]
MRS1097 is a potent antagonist of adenosine hA3 receptor, with the Ki of 100 nM[1]. | [References]
[1] KENNETH A JACOBSON, et al. Pharmacological Characterization of Novel A3 Adenosine Receptor-selective Antagonists. Neuropharmacology. 1997 Sep; 36(9): 1157–1165. |
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