| Identification | Back Directory | [Name]
2-(6-CHLORO-3-PYRIDINYL)-9-AZABICYCLO[4.2.1]NON-2-ENE FUMARATE | [CAS]
200432-86-6 | [Synonyms]
UB 165 FUMARATE
2-(6-CHLORO-3-PYRIDINYL)-9-AZABICYCLO[4.2.1]NON-2-ENE FUMARATE
9-Azabicyclo[4.2.1]non-2-ene, 2-(6-chloro-3-pyridinyl)-, (1R,6R)- | [Molecular Formula]
C13H15ClN2 | [MDL Number]
MFCD06798975 | [MOL File]
200432-86-6.mol | [Molecular Weight]
234.72 |
| Chemical Properties | Back Directory | [Boiling point ]
378.1±37.0 °C(Predicted) | [density ]
1.189±0.06 g/cm3(Predicted) | [storage temp. ]
Desiccate at +4°C | [form ]
Powder | [pka]
9.58±0.40(Predicted) | [Water Solubility ]
Soluble to 100 mM in water with gentle warming |
| Hazard Information | Back Directory | [Uses]
UB 165 Fumarate is a novel presynaptic nicotinic acetylcholine receptor (nAChRs) agonist, which shows immediate potency. | [Biological Activity]
Subtype-selective nicotinic agonist. Full agonist at α 3 β 2- and very weak partial agonist at α 4 β 2- containing nAChRs. K i values are 0.27, 20 (IC 50 ), 2790 and 990 nM for α 4 β 2, α 3, α 7 and α 1 β 1 δ ε respectively. | [storage]
Store at -20°C |
|
|