| Identification | Back Directory | [Name]
L45 | [CAS]
2079885-05-3 | [Synonyms]
L45
LMoses,L Moses
L-Moses >=98% (HPLC)
1,2-Propanediamine, N1,N1-dimethyl-N2-(3-methyl-1,2,4-triazolo[3,4-a]phthalazin-6-yl)-1-phenyl-, (1S,2S)- | [Molecular Formula]
C21H24N6 | [MDL Number]
MFCD31563590 | [MOL File]
2079885-05-3.mol | [Molecular Weight]
360.46 |
| Chemical Properties | Back Directory | [density ]
1.22±0.1 g/cm3(Predicted) | [storage temp. ]
-196°C | [solubility ]
Soluble in DMSO | [form ]
Solid | [pka]
8.00±0.50(Predicted) | [color ]
White to light yellow | [biological source]
Porcine blood |
| Hazard Information | Back Directory | [Uses]
L Moses Dihydrochloride is a potent, selective, and cell-active PCAF bromodomain (Brd) inhibitor. | [in vivo]
L-Moses (L-45) shows no observable cytotoxicity in peripheral blood mononuclear cells (PBMC), good cell-permeability, and metabolic stability in human and mouse liver microsomes, supporting its potential for in vivo use[1]. | [IC 50]
Brd: 126 nM (Kd) | [storage]
Store at -20°C |
|
| Company Name: |
Energy Chemical
|
| Telephone: |
400-0056266 |
| Website: |
www.energy-chemical.com |
|