| Identification | Back Directory | [Name]
Deltasonamide 2
(Deltasonamide2) | [CAS]
2088485-34-9 | [Synonyms]
Deltasonamide 2
Deltasonamide 2
(Deltasonamide2)
1,4-Benzenedisulfonamide, N1-(trans-4-aminocyclohexyl)-N4-[(4-chlorophenyl)methyl]-N4-cyclopentyl-N1-[[2-(methylamino)-4-pyrimidinyl]methyl]- | [Molecular Formula]
C30H39ClN6O4S2 | [MDL Number]
MFCD32062802 | [MOL File]
2088485-34-9.mol | [Molecular Weight]
647.25 |
| Chemical Properties | Back Directory | [Boiling point ]
812.1±75.0 °C(Predicted) | [density ]
1.41±0.1 g/cm3(Predicted) | [storage temp. ]
Store at -20°C | [form ]
Solid | [pka]
10.32±0.70(Predicted) | [color ]
White to off-white |
| Hazard Information | Back Directory | [Uses]
Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM[1]. | [References]
[1] Klein CH, et al. PDEδ inhibition impedes the proliferation and survival of human colorectal cancer cell linesharboring oncogenic KRas. Int J Cancer. 2019 Feb 15;144(4):767-776. DOI:10.1002/ijc.31859 |
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