| Identification | Back Directory | [Name]
BET-IN-2 | [CAS]
2104688-91-5 | [Synonyms]
BET-IN-2
2(1H)-Quinoxalinone, 4-cyclopropyl-6-[[(1S)-1-(2,4-dimethylphenyl)ethyl]amino]-3,4-dihydro-1,3-dimethyl-, (3R)- | [Molecular Formula]
C23H29N3O | [MDL Number]
MFCD31813611 | [MOL File]
2104688-91-5.mol | [Molecular Weight]
363.5 |
| Hazard Information | Back Directory | [Uses]
BET-IN-2 is a BET inhibitor with an IC50 of 52 nM for BRD4-BD1. | [IC 50]
BRD4 BD1: 52 nM (IC50) | [References]
[1] Hu J, et al. Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor. Eur J Med Chem. 2017 Sep 8;137:176-195. DOI:10.1016/j.ejmech.2017.05.049 |
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