| Identification | Back Directory | [Name]
(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE | [CAS]
217480-27-8 | [Synonyms]
818
L-817
L-817,818
L 817,818,L817,818
N2-[[2-(2-Naphthalenyl)-1H-benz[g]indol-3-yl]acetyl-D-lysine(2S)-2-aminopropylester
(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE
D-Lysine, N2-[2-[2-(2-naphthalenyl)-1H-benz[g]indol-3-yl]acetyl]-, (2S)-2-aminopropyl ester | [Molecular Formula]
C33H36N4O3 | [MDL Number]
MFCD09971065 | [MOL File]
217480-27-8.mol | [Molecular Weight]
536.66 |
| Chemical Properties | Back Directory | [Boiling point ]
827.9±65.0 °C(Predicted) | [density ]
1.235±0.06 g/cm3(Predicted) | [storage temp. ]
Store at -20°C | [solubility ]
Soluble to 100 mM in DMSO | [form ]
Powder | [pka]
14.07±0.46(Predicted) | [color ]
White to off-white |
| Hazard Information | Back Directory | [Uses]
L-817,818 is a potent sst5 agonist. | [Biological Activity]
Potent and selective somatostatin sst 5 receptor agonist. K i values are 0.4, 3.3, 52, 64 and 82 nM for cloned human sst 5 , sst 1 , sst 2 , sst 3 and sst 4 receptors respectively. Inhibits growth hormone release from rat pituitary cells (EC 50 = 3.1 nM) and insulin release from mouse pancreatic islets (EC 50 = 0.3 nM) in vitro . | [storage]
Store at -20°C |
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