| Hazard Information | Back Directory | [Uses]
GSK9311 hydrochloride, a less active analogue of GSK6853, can be used as a negative control. GSK9311 hydrochloride inhibits BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively[1]. | [IC 50]
BRPF1: 6.0 (pIC50); BRPF2: 4.3 (pIC50) | [storage]
Store at -20°C | [References]
[1] Bamborough P, et al. GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain. ACS Med Chem Lett. 2016 May 9;7(6):552-7. DOI:10.1021/acsmedchemlett.6b00092 |
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