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2922480-38-2

2922480-38-2 Structure

2922480-38-2 Structure
IdentificationBack Directory
[Name]

L Moses Dihydrochloride
[CAS]

NoCAS
[Synonyms]

L Moses Dihydrochloride
Chemical PropertiesBack Directory
[form ]

Solid
[color ]

White to off-white
Hazard InformationBack Directory
[Uses]

L Moses Dihydrochloride is a potent, selective, and cell-active PCAF bromodomain (Brd) inhibitor.
[in vivo]

L-Moses (L-45) shows no observable cytotoxicity in peripheral blood mononuclear cells (PBMC), good cell-permeability, and metabolic stability in human and mouse liver microsomes, supporting its potential for in vivo use[1].

[IC 50]

Brd: 126 nM (Kd)
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