| Identification | Back Directory | [Name]
Repirinast | [CAS]
73080-51-0 | [Synonyms]
Romet
MY-5116
REPIRINAST
3-Methylbutyl 7,8-dimethyl-4,5-dioxo-6H-pyrano[5,6-c]quinoline-2-carboxylate
Isopentyl 7,8-diMethyl-4,5-dioxo-5,6-dihydro-4H-pyrano[3,2-c]quinoline-2-carboxylate
5，6-Dihydro-7，8-dimethyl-4，5-dioxo-4H-pyrano[3，2-c]quinoline-2-carboxylic acid 3-methylbutyl ester
4H-Pyrano[3,2-c]quinoline-2-carboxylic acid, 5,6-dihydro-7,8-diMethyl-4,5-dioxo-, 3-Methylbutyl Ester | [Molecular Formula]
C20H21NO5 | [MDL Number]
MFCD00867034 | [MOL File]
73080-51-0.mol | [Molecular Weight]
355.38 |
| Chemical Properties | Back Directory | [Melting point ]
236-241° | [Boiling point ]
488.42°C (rough estimate) | [density ]
1.2749 (rough estimate) | [refractive index ]
1.6000 (estimate) | [storage temp. ]
2-8°C | [solubility ]
DMSO (Sparingly, Heated), Methanol (Slightly, Heated) | [form ]
Solid | [pka]
10.09±0.40(Predicted) | [color ]
White to Off-White | [Water Solubility ]
1.2mg/L(temperature not stated) |
| Hazard Information | Back Directory | [Usage]
Antiallergic. | [Description]
Repirinast is an orally-active antiallergic agent useful in the treatment of allergic asthma.
Its activity is reportedly attributed to a metabolite, the corresponding free acid (MY-1250),
which is 17 times more potent than disodium cromoglycate in inhibiting histamine release
due to antigen-antibody reactions. | [Chemical Properties]
Crystallized from chloroform-hexane, melting point 236-241°C. Acute toxicity LD50 in mice, rats, rabbits and dogs (mg/kg): >5000 oral. | [Originator]
Mitsubishi (Japan) | [Uses]
Antiallergic. | [Definition]
ChEBI: Repirinast is an organic molecular entity. | [Brand name]
Romet |
|
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J & K SCIENTIFIC LTD.
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NCE Biomedical Co.,Ltd.
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