| Identification | Back Directory | [Name]
D-VAL-PHE-LYS CHLOROMETHYL KETONE, DIHYDROCHLORIDE | [CAS]
75590-17-9 | [Synonyms]
DVal-Phe-Lys-CMK
PLASMIN INHIBITOR, 2HCL
valyl-phenylalanyl-lysine chloromethyl ketone
D-VAL-PHE-LYS CHLOROMETHYL KETONE, DIHYDROCHLORIDE
L-Phenylalaninamide, D-valyl-N-[(1S)-5-amino-1-(2-chloroacetyl)pentyl]- | [Molecular Formula]
C21H33ClN4O3 | [MDL Number]
MFCD00077405 | [MOL File]
75590-17-9.mol | [Molecular Weight]
424.96 |
| Chemical Properties | Back Directory | [Boiling point ]
707.0±60.0 °C(Predicted) | [density ]
1.160±0.06 g/cm3(Predicted) | [storage temp. ]
2-8°C | [solubility ]
DMSO: 5mg/mL | [form ]
lyophilized solid | [pka]
13.06±0.46(Predicted) | [color ]
off-white | [Sequence]
{d-Val}-Phe-Lys-{CMK} |
| Hazard Information | Back Directory | [Uses]
D-Val-Phe-Lys-CMK (D-Val-Phe-Lys Chloromethyl ketone) can inhibit plasmin activity[1]. | [Biological Activity]
Cell permeable: no''Primary Target
Human plasmin''Product does not compete with ATP.''Reversible: no''Target IC50: 100 pM for human plasmin | [References]
[1] F Laube, et al. Cell surface antigens in renal tumour cells: detection by immunoluminescence and enzymatic analysis. Br J Cancer. 2001 Sep 14;85(6):924-9. DOI:10.1054/bjoc.2001.2004 |
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YantaiBio
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13758194781; 13758194781 |
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