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757176-96-8

757176-96-8 Structure

757176-96-8 Structure
IdentificationBack Directory
[Name]

1,2,3,11b-Tetrahydro[1]benzopyrano[4,3,2-de]isoquinoline-8,9-diol
[CAS]

757176-96-8
[Synonyms]

Dinoxyline
[Molecular Formula]

C15H13NO3
[MOL File]

757176-96-8.mol
[Molecular Weight]

255.27
Chemical PropertiesBack Directory
[Boiling point ]

448.0±45.0 °C(Predicted)
[density ]

1.405±0.06 g/cm3(Temp: 20 °C; Press: 760 Torr)(Predicted)
[pka]

8.98±0.20(Predicted)
Hazard InformationBack Directory
[Uses]

Dinoxyline is a potent agonist at dopamine receptors (Ki = 7 nM, 6 nM, 5 nM, 43 nM for D1, D2, D3 and D4). Dinoxyline can be utilized in neurological research[1].
[References]

[1] Fowler JC, et al. Receptor conformations involved in dopamine D(2L) receptor functional selectivity induced by selected transmembrane-5 serine mutations. Mol Pharmacol. 2012 Jun;81(6):820-31. DOI:10.1124/mol.111.075457
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