| Identification | Back Directory | [Name]
SAM-531 | [CAS]
925448-93-7 | [Synonyms]
SAM-531
WAY-262
PF05212365
PF-05212365
WAY-262,531
P -05212365
Cerlapirdine
N,N-Dimethyl-3-[[3-(1-naphthalenylsulfonyl)-1H-indazol-5-yl]oxy]-1-propanamine
1-Propanamine, N,N-dimethyl-3-[[3-(1-naphthalenylsulfonyl)-1H-indazol-5-yl]oxy]-
antagonist,inhibit,5-HT Receptor,5-hydroxytryptamine,5-HT6,oral,Cerlapirdine,PF 05212365,selective,Alzheimer's disease,Serotonin Receptor,5-hydroxytryptamine Receptor,Inhibitor | [Molecular Formula]
C22H23N3O3S | [MDL Number]
MFCD18782738 | [MOL File]
925448-93-7.mol | [Molecular Weight]
409.5 |
| Chemical Properties | Back Directory | [Boiling point ]
662.9±45.0 °C(Predicted) | [density ]
1.300±0.06 g/cm3(Predicted) | [storage temp. ]
4°C, protect from light | [solubility ]
DMSO : 41.67 mg/mL (101.76 mM; ultrasonic and warming and adjust pH to 3 with HCl and heat to 60°C) | [form ]
Solid | [pka]
9.70±0.40(Predicted) | [color ]
Off-white to yellow |
| Hazard Information | Back Directory | [Uses]
Cerlapirdine is a selective and potent full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor (1). Used in the symptomatic treatment of Alzheimer’s disease. | [IC 50]
5-HT6 Receptor |
|
| Company Name: |
Energy Chemical
|
| Tel: |
021-58432009 400-005-6266 |
| Website: |
http://www.energy-chemical.com |
|