YAP-TEAD Inhibitor 1
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- CAS号:
- 1659305-78-8
- 英文名:
- YAP-TEAD Inhibitor 1
- 英文别名:
- YAP-TEAD-IN-1;Y413924] YAP-TEAD;YAP-TEAD Inhibitor 1;YAP-TEAD-IN-1 (Peptide 17);YAP-TEAD Inhibitor 1 (Peptide 17) ，S8164;L-α-Glutamine, N-acetyl-L-valyl-L-prolyl-3-chloro-L-phenylalanyl-L-homocysteinyl-L-leucyl-L-arginyl-L-lysyl-L-norleucyl-L-prolyl-L-alanyl-L-seryl-L-phenylalanyl-L-cysteinyl-L-lysyl-L-prolyl-L-prolyl-, cyclic (4→13)-disulfide
- 中文名:
- YAP-TEAD Inhibitor 1
- 中文别名:
- YAP-TEAD抑制剂1(肽17)TFA;竞争性肽类抑制剂YAP-TEAD-IN-1;Y413924] YAP-TEAD抑制剂1(肽17)TFA;YAP-TEAD Inhibitor 1 (Peptide 17) ,S8164;AC-VAL-PRO-PHE(3-CL)-HOMOCYS-LEU-ARG-LYS-NLE-PRO-ALA-SER-PHE-CYS-LYS-PRO-PRO-GLU-NH2 (DISULFIDE BRIDGE:HCY4-CYS13)
- CBNumber:
- CB24656621
- 分子式:
- C93H144ClN23O21S2
- 分子量:
- 2019.86
- MOL File:
- 1659305-78-8.mol
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YAP-TEAD Inhibitor 1化学性质
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密度:
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1.45±0.1 g/cm3(Predicted)
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储存条件:
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Store at -20°C
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形态:
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Solid
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酸度系数(pKa):
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4.45±0.10(Predicted)
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颜色:
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White to off-white
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水溶解性:
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Water: 40 mg/mL (19.80 mM);
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YAP-TEAD Inhibitor 1性质、用途与生产工艺
YAP-TEAD-IN-1 是 YAP–TEAD 相互作用的有效的竞争性肽类抑制剂 (IC50=25 nM)。YAP-TEAD-IN-1 是一种 17mer 的多肽，与 YAP (50-171) (Kd=40 nM) 相比，其与 TEAD1 的结合亲和力更高 (Kd=15 nM)。
YAP-TEAD Inhibitor 1
上下游产品信息
上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
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| 2025/09/19 | S8164 | YAP-TEAD Inhibitor 1
YAP-TEAD Inhibitor 1 (Peptide 17) | 1659305-78-8 | 1mg | 1613.48元 |
| 2025/09/19 | S8164 | YAP-TEAD Inhibitor 1 (Peptide 17) | 1659305-78-8 | 5mg | 5708.64元 |
YAP-TEAD Inhibitor 1
生产厂家
1659305-78-8, YAP-TEAD Inhibitor 1 相关搜索:
- 目录肽
- 药靶配体
- 多肽-目录肽
- C93H144ClN23O21S2
- YAP-TEAD Inhibitor 1 (Peptide 17) ,S8164
- 竞争性肽类抑制剂YAP-TEAD-IN-1
- YAP-TEAD抑制剂1(肽17)TFA
- Y413924] YAP-TEAD抑制剂1(肽17)TFA
- AC-VAL-PRO-PHE(3-CL)-HOMOCYS-LEU-ARG-LYS-NLE-PRO-ALA-SER-PHE-CYS-LYS-PRO-PRO-GLU-NH2 (DISULFIDE BRIDGE:HCY4-CYS13)
- 1659305-78-8
- YAP-TEAD Inhibitor 1 (Peptide 17) ，S8164
- YAP-TEAD-IN-1 (Peptide 17)
- Y413924] YAP-TEAD
- L-α-Glutamine, N-acetyl-L-valyl-L-prolyl-3-chloro-L-phenylalanyl-L-homocysteinyl-L-leucyl-L-arginyl-L-lysyl-L-norleucyl-L-prolyl-L-alanyl-L-seryl-L-phenylalanyl-L-cysteinyl-L-lysyl-L-prolyl-L-prolyl-, cyclic (4→13)-disulfide
- YAP-TEAD-IN-1
- YAP-TEAD Inhibitor 1