ENPP1 Inhibitor C
- CAS No.
- 2378640-92-5
- Chemical Name:
- ENPP1 Inhibitor C
- Synonyms
- Enpp-1-IN-2;ENPP1 Inhibitor C;6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine;[1,2,4]Triazolo[1,5-a]pyrimidin-7-amine, 6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-
- CBNumber:
- CB06197878
- Molecular Formula:
- C15H18N6
- Molecular Weight:
- 282.34
- MDL Number:
- MOL File:
- 2378640-92-5.mol
- MSDS File:
- SDS
- TDS File:
- TDS
ENPP1 Inhibitor C price
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Cayman Chemical | 29809 | ENPP1 Inhibitor C ≥98% | 2378640-92-5 | 1mg | $95 | 2026-04-30 | Buy |
| Cayman Chemical | 29809 | ENPP1 Inhibitor C ≥98% | 2378640-92-5 | 5mg | $417 | 2026-04-30 | Buy |
| Cayman Chemical | 29809 | ENPP1 Inhibitor C ≥98% | 2378640-92-5 | 10mg | $692 | 2026-04-30 | Buy |
| Biosynth | DVD64092 | Enpp1 inhibitor C | 2378640-92-5 | 10mg | $1009 | 2026-06-04 | Buy |
| Biosynth | DVD64092 | Enpp1 inhibitor C | 2378640-92-5 | 25mg | $1645.25 | 2026-06-04 | Buy |
ENPP1 Inhibitor C Chemical Properties, Uses, Production
Description
ENPP1 inhibitor C is an inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1; IC50 = 0.26 μM in a cell-free assay).1 It is selective for ENPP1 over ENPP2-7 at 10 μM. ENPP1 inhibitor C decreases ENPP1 activity in MDA-MB-231 human breast and C6 rat glioma cancer cells when used at a concentration of 10 μM.
Uses
Enpp-1-IN-2 (Compound C) is a potent ENPP1 (ectonucleotide pyrophosphatase/phosphodiesterase 1) inhibitor with IC50 values of 0.26, 0.48 and 2.0 μM evaluated by means of TG-mAMP, pNP-TMP, and ATP assays, respectively. TG (Tokyo Green)-mAMP: a newly synthesized sensitive ENPP1 fluorescence probe[1].
References
1. Kawaguchi, M., Han, X., Hisada, T., et al. Development of an ENPP1 fluorescence probe for inhibitor screening, cellular imaging, and prognostic assessment of malignant breast cancer J. Med. Chem. 62(20),9254-9269(2019).
ENPP1 Inhibitor C Preparation Products And Raw materials
Raw materials
Preparation Products
ENPP1 Inhibitor C Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Shanghai Beckham Medical Technology Co., Ltd | 13816613772 | huahero21@sina.com | China | 2996 | 55 |
| Shanghai EFE Biological Technology Co., Ltd. | 021-65675885 18964387627 | info@efebio.com | China | 9799 | 58 |
| Shanghai Chaolan Chemical Technology Center | QQ：65489617 13301690235 | Sales@ATKchemical.com | China | 9699 | 58 |
| Shenzhen SUNGENING Bio-Medical Co., Ltd. | 0755-28967200 13631290199 | wxf@sungening.com | China | 9609 | 60 |
| Shanghai Hongye Biotechnology Co. Ltd | 400-9205774 400-920-5774 | sales@glpbio.cn | China | 6705 | 58 |
| ChemeGen(Shanghai) Biotechnology Co.,Ltd. | 18818260767 | sales@chemegen.com | China | 11123 | 58 |
| Wuhan Topule | +86-02787215551 19945035818 | 2936752263@qq.com | China | 7983 | 58 |
| TargetMol Chemicals Inc. | 4008200310 15002144251 | marketing@tsbiochem.com | China | 24951 | 58 |
| Xianning Shen Lan Biomedical Research and Development Co., Ltd. | 18171815831 | 1341138380@qq.com | China | 4573 | 58 |
| Shanghai Tachizaki Biomedical Research Center | 18014399201 | sales@chemlab-tachizaki.com | China | 2934 | 58 |
