ChemicalBook >> CAS DataBase List >>GSK5959
GSK5959
- CAS No.
- 901245-65-6
- Chemical Name:
- GSK5959
- Synonyms
- CS-1636;GSK5959;BRPF1-IN-3;GSK 5959 ，S5916;GSK-5959;GSK5959;GSK-5959, 10 mM in DMSO;N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide;Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxy-;N-(1,3-dimethyl-2-oxo-6-(piperidin-1-yl)-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methoxybenzamide;BRPF3,GSK5959,bromodomain,Inhibitor,inhibit,BRD1,BRPF1,Epigenetic Reader Domain,GSK-5959,GSK 5959,BRPF2,epigenetics
- CBNumber:
- CB23040788
- Molecular Formula:
- C22H26N4O3
- Molecular Weight:
- 394.47
- MDL Number:
- MFCD14744183
- MOL File:
- 901245-65-6.mol
Last updated:2025-10-13 11:45:57
| Product description | Number | Pack Size | Price |
| GSK5959 ≥98% | 18123 | 1mg | $32 |
| GSK5959 ≥98% | 18123 | 5mg | $100 |
| GSK5959 ≥98% | 18123 | 10mg | $184 |
| GSK5959 ≥98% | 18123 | 25mg | $381 |
| GSK5959 ≥99%(HPLC) | 5385 | 10 | $159 |
| More product size | |||
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS07 |
|---|---|
| Signal word | Warning |
| Hazard statements | H302-H315-H319-H335 |
| Precautionary statements | P261-P305+P351+P338 |
GSK5959 price More Price(22)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Cayman Chemical | 18123 | GSK5959 ≥98% | 901245-65-6 | 1mg | $32 | 2024-03-01 | Buy |
| Cayman Chemical | 18123 | GSK5959 ≥98% | 901245-65-6 | 5mg | $100 | 2024-03-01 | Buy |
| Cayman Chemical | 18123 | GSK5959 ≥98% | 901245-65-6 | 10mg | $184 | 2024-03-01 | Buy |
| Cayman Chemical | 18123 | GSK5959 ≥98% | 901245-65-6 | 25mg | $381 | 2024-03-01 | Buy |
| Tocris | 5385 | GSK5959 ≥99%(HPLC) | 901245-65-6 | 10 | $159 | 2021-12-16 | Buy |
GSK5959 Chemical Properties,Uses,Production
Description
GSK 5959 exhibits >100-fold selectivity for BRPF1 (IC50 = 80 nM) over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3, which is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.
Uses
GSK5959 is as elective BRPF1 bromodomain inhibitor.
storage
Store at +4°C
GSK5959 Preparation Products And Raw materials
Raw materials
Preparation Products
Global( 81)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| ATK CHEMICAL COMPANY LIMITED | +undefined-21-51877795 | ivan@atkchemical.com | China | 33024 | 60 |
| TargetMol Chemicals Inc. | +1-781-999-5354; +17819995354 | marketing@targetmol.com | United States | 32434 | 58 |
| Career Henan Chemica Co | +86-0371-86658258 +8613203830695 | laboratory@coreychem.com | China | 30229 | 58 |
| InvivoChem | +1-708-310-1919 +1-13798911105 | sales@invivochem.cn | United States | 6391 | 58 |
| Nanjing Doge Biomedical Technology Co., Ltd | +86-25-58227606 +86-15305155328 | sales@dogechemical.com | China | 4128 | 58 |
| ShenZhen Trendseen Biological Technology Co.,Ltd. | 13417589054 | trendseenbio@gmail.com | China | 11681 | 58 |
| HANGZHOU LEAP CHEM CO., LTD. | +86-571-87711850 | market18@leapchem.com | China | 43339 | 58 |
| Jilin Chinese Academy of Sciences-yanshen Technology | +undefined18143011203 | info@chemextension.com | China | 42056 | 58 |
| Aladdin Scientific | tp@aladdinsci.com | United States | 57505 | 58 | |
| Amadis Chemical Company Limited | 571-89925085 | sales@amadischem.com | China | 131957 | 58 |
GSK5959
BRPF1-IN-3
N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide
GSK-5959;GSK5959
CS-1636
Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxy-
BRPF3,GSK5959,bromodomain,Inhibitor,inhibit,BRD1,BRPF1,Epigenetic Reader Domain,GSK-5959,GSK 5959,BRPF2,epigenetics
N-(1,3-dimethyl-2-oxo-6-(piperidin-1-yl)-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methoxybenzamide
GSK-5959, 10 mM in DMSO
GSK 5959 ，S5916
901245-65-6
Inhibitors
