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ChemicalBook >> CAS DataBase List >>(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester Structure
(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester structure
CAS No.
1256756-88-3
Chemical Name:
(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester
Synonyms
SP-2086;CPDA1089;RETAGLIPTIN; SP-2086;RetagliptinPhosphate;Triazolam Impurity 8;Reagliptin (phosphate);Retagliptin Phosphate, 10 mM in DMSO;SP-2086,Retagliptin Phosphate,DPP-4,SP2086,inhibit,GLP-1,T2DM,Retagliptin,DPP,Inhibitor,Dipeptidyl Peptidase;methyl (R)-7-(3-amino-4-(2,4,5-trifluorophenyl)butanoyl)-3-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylate phosphate;(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester
CBNumber:
CB23121243
Molecular Formula:
C19H18F6N4O3
Molecular Weight:
464.3616392
MDL Number:
MFCD31692418
MOL File:
1256756-88-3.mol
Last updated:2025-09-23 08:43:30
Request For Quotation

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester Properties

storage temp. Store at -20°C
solubility DMSO : ≥ 150 mg/mL (266.73 mM)
form Solid
color White to light yellow
FDA UNII 24NZ3UE3DJ

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
ChemScene CS-0059159 Retagliptin(phosphate) 99.89% 1256756-88-3 5mg $150 2021-12-16 Buy
ChemScene CS-0059159 Retagliptin(phosphate) 99.89% 1256756-88-3 10mg $240 2021-12-16 Buy
ChemScene CS-0059159 Retagliptin(phosphate) 99.89% 1256756-88-3 50mg $750 2021-12-16 Buy
ChemScene CS-0059159 Retagliptin(phosphate) 99.89% 1256756-88-3 100mg $1200 2021-12-16 Buy
Chemenu CM328796 methyl7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-3-(trifluoromethyl)-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-1-carboxylate;phosphoricacid 95%+ 1256756-88-3 5g $2208 2021-12-16 Buy
Product number Packaging Price Buy
CS-0059159 5mg $150 Buy
CS-0059159 10mg $240 Buy
CS-0059159 50mg $750 Buy
CS-0059159 100mg $1200 Buy
CM328796 5g $2208 Buy

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester Chemical Properties,Uses,Production

Uses

Retagliptin phosphate (SP2086 phosphate) is a selective, competitive and orally active dipeptidyl peptidase-4 (DPP-4) inhibitor. Retagliptin phosphate can be used for type 2 diabetes mellitus (T2DM) research[1].

IC 50

DPP-4

References

[1] Hu C, et al. Pharmacokinetics of Phosphate Retagliptin Tabletin in Patients with Renal Dysfunction. Sichuan Da Xue Xue Bao Yi Xue Ban. 2018 Jan;49(1):74-80. PMID:29737094
[2] Avivit Cahn, et al. An update on DPP-4 inhibitors in the management of type 2 diabetes. Expert Opin Emerg Drugs. 2016 Dec;21(4):409-419. DOI:10.1080/14728214.2016.1257608

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester Preparation Products And Raw materials

Raw materials

Preparation Products

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester Suppliers

Global( 23)Suppliers
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc. 		+1-781-999-5354; +17819995354 marketing@targetmol.com United States 32432 58
TargetMol Chemicals Inc. 		+1-781-999-5354; support@targetmol.com United States 39031 58
Tianjin Yao Technology Development Co., Ltd. 022-18902014291 18902014291 byswxsb01@163.com China 101 58
ShangHai Caerulum Pharma Discovery Co., Ltd. 18149758185 sales-cpd@caerulumpharma.com China 3503 58
Sichuan Wei Keqi Biological Technology Co., Ltd. 028-81700200 18116577057 3003855609@qq.com China 7781 56
Jinan Yaoyan Pharmaceutical Co., Ltd. jnyaoyan@163.com China 3069 58
Nanjing Meihao Pharmaceutical Technology Co., Ltd. meitaochem@126.com meitaochem@126.com China 19103 58
ChemeGen(Shanghai) Biotechnology Co.,Ltd. 18818260767 sales@chemegen.com China 11218 58
Guangzhou Younan Technology Co., Ltd 020-82000279 18988968278 YN_research@163.com China 3003 58
TargetMol Chemicals Inc. 4008200310 marketing@tsbiochem.com China 24989 58
Supplier Advantage
TargetMol Chemicals Inc. 		58
TargetMol Chemicals Inc. 		58
Tianjin Yao Technology Development Co., Ltd. 58
ShangHai Caerulum Pharma Discovery Co., Ltd. 58
Sichuan Wei Keqi Biological Technology Co., Ltd. 56
Jinan Yaoyan Pharmaceutical Co., Ltd. 58
Nanjing Meihao Pharmaceutical Technology Co., Ltd. 58
ChemeGen(Shanghai) Biotechnology Co.,Ltd. 58
Guangzhou Younan Technology Co., Ltd 58
TargetMol Chemicals Inc. 58

View Lastest Price from (R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
Retagliptin Phosphate pictures 2025-09-22 Retagliptin Phosphate
1256756-88-3
 US $30.00-58.00 / mg 98.97% 10g TargetMol Chemicals Inc.
Retagliptin Phosphate pictures 2025-09-22 Retagliptin Phosphate
1256756-88-3
 US $30.00-58.00 / mg 98.97% 10g TargetMol Chemicals Inc.

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester Spectrum

(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester(1256756-88-3)1HNMR
(R)-7-[3-amino-4-(2,4,5-trifluoro-phenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1- carboxylic acid methyl ester CPDA1089 RetagliptinPhosphate RETAGLIPTIN; SP-2086 SP-2086 methyl (R)-7-(3-amino-4-(2,4,5-trifluorophenyl)butanoyl)-3-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylate phosphate SP-2086,Retagliptin Phosphate,DPP-4,SP2086,inhibit,GLP-1,T2DM,Retagliptin,DPP,Inhibitor,Dipeptidyl Peptidase Reagliptin (phosphate) Triazolam Impurity 8 Retagliptin Phosphate, 10 mM in DMSO 1256756-88-3