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5-METHOXYGRAMINE

5-METHOXYGRAMINE structure

CAS No.: 16620-52-3

Chemical Name:: 5-METHOXYGRAMINE

Synonyms: NSC 88885;methoxygramine;5-METHOXYGRAMINE;TIMTEC-BB SBB003509;5-METHOXYGRAMINE 99%;5-Methoxygramine,99%;3-ETHYL-1H-PYRAZOL-5-AMINE HCL;2-dimethylaminomethyl-5-methoxyindole;5-methoxy-3-(dimethylaminomethyl)indole;3-(DIMETHYLAMINOMETHYL)-5-METHOXY-INDOLE

CBNumber:: CB5245525

Molecular Formula:: C12H16N2O

Molecular Weight:: 204.27

MDL Number:: MFCD00005630

MOL File:: 16620-52-3.mol

MSDS File:: SDS

TDS File:: TDS

Last updated:2026-04-24 14:58:19

Product description	Number	Pack Size	Price
5-Methoxygramine 99%	M14870	5g	$225
5-Methoxygramine	M263278	10mg	$45
N-[(5-Methoxy-1H-indol-3-yl)methyl]-N,N-dimethylamine	Y7751	1g	$104
5-METHOXYGRAMINE 95.00%	CHM0031161	1G	$654.89
5-METHOXYGRAMINE 95.00%	CHM0031161	5G	$970.2
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5-METHOXYGRAMINE Properties

Melting point	123-126 °C (lit.)
Boiling point	342.77°C (rough estimate)
Density	1.0565 (rough estimate)
refractive index	1.6000 (estimate)
storage temp.	Refrigerator (+4°C)
pka	16.70±0.30(Predicted)
BRN	170533
InChI	1S/C12H16N2O/c1-14(2)8-9-7-13-12-5-4-10(15-3)6-11(9)12/h4-7,13H,8H2,1-3H3
InChIKey	GOERTRUXQHDLHC-UHFFFAOYSA-N
SMILES	COc1ccc2[nH]cc(CN(C)C)c2c1
CAS DataBase Reference	16620-52-3(CAS DataBase Reference)
FDA UNII	J6ZN008RY8
UNSPSC Code	12352100
NACRES	NA.22

SAFETY

Risk and Safety Statements

Symbol(GHS)	GHS07,GHS05
Signal word	Danger
Hazard statements	H302-H314
Precautionary statements	P264-P270-P301+P312-P330-P501-P260-P264-P280-P301+P330+P331-P303+P361+P353-P363-P304+P340-P310-P321-P305+P351+P338-P405-P501
PPE	Eyeshields, Gloves, type N95 (US)
Hazard Codes	C,Xi
Risk Statements	34-22
Safety Statements	22-24/25
WGK Germany	3
RTECS	NL7700000
F	10
HS Code	29339900
Storage Class	11 - Combustible Solids
Toxicity	mouse,LD50,intraperitoneal,130mg/kg (130mg/kg),Psychopharmacologia Vol. 16, Pg. 385, 1970.

5-METHOXYGRAMINE price More Price(15)

Manufacturer	Product number	Product description	CAS number	Packaging	Price	Updated	Buy
Sigma-Aldrich	M14870	5-Methoxygramine 99%	16620-52-3	5g	$225	2023-06-20	Buy
TRC	M263278	5-Methoxygramine	16620-52-3	10mg	$45	2021-12-16	Buy
AK Scientific	Y7751	N-[(5-Methoxy-1H-indol-3-yl)methyl]-N,N-dimethylamine	16620-52-3	1g	$104	2021-12-16	Buy
American Custom Chemicals Corporation	CHM0031161	5-METHOXYGRAMINE 95.00%	16620-52-3	1G	$654.89	2021-12-16	Buy
American Custom Chemicals Corporation	CHM0031161	5-METHOXYGRAMINE 95.00%	16620-52-3	5G	$970.2	2021-12-16	Buy

Product number	Packaging	Price	Buy
M14870	5g	$225	Buy
M263278	10mg	$45	Buy
Y7751	1g	$104	Buy
CHM0031161	1G	$654.89	Buy
CHM0031161	5G	$970.2	Buy

5-METHOXYGRAMINE Chemical Properties,Uses,Production

Chemical Properties

white to almost white crystalline powder

Uses

• ;Reactant for preparation of dopamine D2 receptor antagonists1• ;Reactant for asymmetric preparation of ethenyl(tetrahydro)carbazoledicarboxylates via gold(I)-catalyzed intramolecular Friedel-Crafts allylic alkylation reaction2• ;Reactant for preparation of N-substituted 3-aryl-8-azabicyclo[3.2.1]octan-3-ols as dopamine D2-like receptor ligands3• ;Reactant for preparation of substituted N-trimethoxybenzoyl indoles, indolines, and a tetrahydroquinoline via N-aroylation with trimethoxybenzoyl chloride or anhydride as antitubulin agents4• ;Reactant for preparation of in

Uses

Reactant for preparation of dopamine D2 receptor antagonists
Reactant for asymmetric preparation of ethenyl(tetrahydro)carbazoledicarboxylates via gold(I)-catalyzed intramolecular Friedel-Crafts allylic alkylation reaction
Reactant for preparation of N-substituted 3-aryl-8-azabicyclo[3.2.1]octan-3-ols as dopamine D2-like receptor ligands
Reactant for preparation of substituted N-trimethoxybenzoyl indoles, indolines, and a tetrahydroquinoline via N-aroylation with trimethoxybenzoyl chloride or anhydride as antitubulin agents
Reactant for preparation of indolylmethanesulfonamide and its methoxy derivatives

5-METHOXYGRAMINE Preparation Products And Raw materials

Raw materials

5-Methoxyindole Formaldehyde Diethyl ether Hydrochloric acid Acetic acid

Sodium hydroxide Dimethylamine

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Preparation Products

5-METHOXYGRAMINE Suppliers

Global( 69)Suppliers

Supplier	Tel	Email	Country	ProdList	Advantage
Alchem Pharmtech,Inc.	8485655694	sales@alchempharmtech.com	United States	63687	58
CONIER CHEM AND PHARMA LIMITED	+8618523575427	sales@conier.com	China	49977	58
Dayang Chem (Hangzhou) Co.,Ltd.	+86-0571-88938639 +8617705817739	info@dycnchem.com	China	52705	58
GIHI CHEMICALS CO.,LIMITED	+86-571-86217390; +8618058761490	info@gihichemicals.com	China	49968	58
Nanjing Bicbiotechnology Co., Ltd	+86-2552131256 +86-18251840740	sales@bicbiotech.com	China	5994	58
Aladdin Scientific		tp@aladdinsci.com	United States	57505	58
Amadis Chemical Company Limited	571-89925085	sales@amadischem.com	China	131957	58
Mainchem Co., Ltd.	+86-0592-6210733	sale@mainchem.com	China	32343	55
Chemwill Asia Co.,Ltd.	86-21-51086038	chemwill_asia@126.com	CHINA	23912	58
J & K SCIENTIFIC LTD.	18210857532; 18210857532	jkinfo@jkchemical.com	China	96815	76

Supplier	Advantage
Alchem Pharmtech,Inc.	58
CONIER CHEM AND PHARMA LIMITED	58
Dayang Chem (Hangzhou) Co.,Ltd.	58
GIHI CHEMICALS CO.,LIMITED	58
Nanjing Bicbiotechnology Co., Ltd	58
Aladdin Scientific	58
Amadis Chemical Company Limited	58
Mainchem Co., Ltd.	55
Chemwill Asia Co.,Ltd.	58
J & K SCIENTIFIC LTD.	76

5-METHOXYGRAMINE Spectrum

5-METHOXYGRAMINE(16620-52-3)¹HNMR 5-METHOXYGRAMINE(16620-52-3)Raman 5-METHOXYGRAMINE(16620-52-3)IR

16620-52-3(5-METHOXYGRAMINE)Related Search:

Gramine 4-Methoxygramine 6-METHOXYGRAMINE 5-BENZYLOXYGRAMINE 3-DIMETHYLAMINOMETHYL-5-METHOXY-1H-INDOLE-2-CARBOXYLIC ACID ETHYL ESTER

2-ACETYL-8-TRIFLUOROMETHOXY-2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLE (5-METHOXY-1H-INDOL-3-YL)(PIPERIDINO)METHANETHIONE Oxybis((5,3-indolylene)methylene)bis(trimethylammonium) bis(methyl sul fate) 5-METHOXY-2-METHYLGRAMINE 5-ETHYL-2-(5-METHOXY-1H-INDOL-3-YL)-7-METHYL-1,3-DIAZATRICYCLO[3.3.1.1~3,7~]DECAN-6-ONE

5-METHOXYGRAMINE 8-BENZYLOXY-2-METHYL-2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLE AKOS JY2083007 2-ACETYL-8-METHOXY-2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLE 1-[(5-methoxy-1H-indol-3-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxylic acid

AKOS JY2083279

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5-METHOXYGRAMINE 99% 5-Methoxygramine, N,N-Dimethyl-(5-methoxy-1H-indol-3-yl)methylamine methoxygramine 5-Methoxygramine or 5-Methoxy-3-(Dimethylaminomethyl)-indole (5-methoxy-1H-indol-3-yl)methyl-dimethylammonium 3-ETHYL-1H-PYRAZOL-5-AMINE HCL 5-Methoxygramine,99% NSC 88885 3-((dimethylamino)methyl)-5-methoxy-indol 5-methoxy-3-(dimethylaminomethyl)indole 5-methoxy-n,n-dimethyl-1h-indole-3-methanamin TIMTEC-BB SBB003509 3-[(Dimethylamino)methyl]-5-methoxy-1H-indole 3-(DIMETHYLAMINOMETHYL)-5-METHOXY-INDOLE (5-METHOXY-1H-INDOL-3-YLMETHYL)-DIMETHYL-AMINE 5-METHOXYGRAMINE 2-dimethylaminomethyl-5-methoxyindole N-[(5-METHOXY-1H-INDOL-3-YL)METHYL]-N,N-DIMETHYLAMINE 1H-Indole-3-methanamine, 5-methoxy-N,N-dimethyl- 5-Methoxy-N,N-dimethyl-1H-indole-3-methanamine 16620-52-3 Heterocyclic Building Blocks Indoles Building Blocks Building Blocks C12 Chemical Synthesis Heterocyclic Building Blocks Indoles Indoline & Oxindole Heterocyclic Compounds Indoles and derivatives