PKC-theta inhibitor 1
- CAS No.
- 1160501-81-4
- Chemical Name:
- PKC-theta inhibitor 1
- Synonyms
- PKCθ inhibitor 22;PKC-theta inhibitor 1;PKCtheta inhibitor 1,PKC theta inhibitor 1;3-Oxetanemethanamine, 3-[3-[3-(trifluoromethyl)-1H-pyrazolo[3,4-b]pyridin-4-yl]phenyl]-
- CBNumber:
- CB75821322
- Molecular Formula:
- C17H15F3N4O
- Molecular Weight:
- 348.32
- MDL Number:
- MFCD32201103
- MOL File:
- 1160501-81-4.mol
- MSDS File:
- SDS
PKC-theta inhibitor 1 price
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| ChemScene | CS-0102613 | PKC-theta inhibitor 1 99.45% | 1160501-81-4 | 1mg | $342 | 2026-06-04 | Buy |
| ChemScene | CS-0102613 | PKC-theta inhibitor 1 99.45% | 1160501-81-4 | 5mg | $1029 | 2026-06-04 | Buy |
| aablocks | AA01WJCP | PKC-theta inhibitor 1 >98% | 1160501-81-4 | 1mg | $387 | 2026-06-01 | Buy |
| aablocks | AA01WJCP | PKC-theta inhibitor 1 >98% | 1160501-81-4 | 5mg | $1091 | 2026-06-01 | Buy |
PKC-theta inhibitor 1 Chemical Properties, Uses, Production
Uses
PKC-theta inhibitor 1 is the PKCθ inhibitor with an Ki value of 6 nM, inhibits IL-2 production in vivo with an IC50 of 0.19 μM. PKC-theta inhibitor 1 demonstrates a reduction of symptoms in a mouse model of multiple sclerosis[1].
IC 50
PKCθ: 6 nM (Ki); PKCδ: 392 μM (Ki); PKCα: 1020 μM (Ki); IL-2 production: 0.19 μM (IC50)
References
[1] Collier PN, et al. Discovery of Selective, Orally Bioavailable Pyrazolopyridine Inhibitors of Protein Kinase Cθ (PKCθ) That Ameliorate Symptoms of Experimental Autoimmune Encephalomyelitis. ACS Med Chem Lett. 2019 Jun 27;10(8):1134-1139. DOI:10.1021/acsmedchemlett.9b00134
PKC-theta inhibitor 1 Preparation Products And Raw materials
Raw materials
Preparation Products
PKC-theta inhibitor 1 Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| BOC Sciences | 1-631-485-4226; 16314854226 | info@bocsci.com | United States | 9920 | 65 |
| Sichuan Wei Keqi Biological Technology Co., Ltd. | 028-81700200 18116577057 | 3003855609@qq.com | China | 7717 | 56 |
| Fan De(Beijing) Biotechnology Co., Ltd. | 15911056312 | liming@bio-fount.com | China | 9718 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; +1-00000000000 | marketing@targetmol.com | United States | 32431 | 58 |
| TargetMol Chemicals Inc. | 4008200310 15002144251 | marketing@tsbiochem.com | China | 24951 | 58 |
| Suzhou Haiben Pharmaceutical Co., Ltd | 19353112242 | 1816280386@qq.com | China | 8041 | 58 |
| Shandong Dayou Pharmaceutical Research and Development Co., Ltd. | hanfangpharma@126.com 15165037910 | hanfangpharma@126.com | China | 25800 | 58 |
| RD International Technology Co., Limited | 18024082417 | market@ubiochem.com | China | 9831 | 58 |
| TargetMol Chemicals Inc. | 13564774135 | marketing@targetmol.com | United States | 19950 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; | support@targetmol.com | United States | 38999 | 58 |
View Latest Price from PKC-theta inhibitor 1 manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2026-04-20 | PKC-theta inhibitor 1
1160501-81-4
|
$1820.00-3100.00 | 10g | TargetMol Chemicals Inc. | |||
 |
2025-08-22 | PKC-theta inhibitor 1
1160501-81-4
|
$1820.00-3100.00 | 10g | TargetMol Chemicals Inc. |
-
- PKC-theta inhibitor 1
1160501-81-4
- $1820.00-3100.00
- TargetMol Chemicals Inc.
-
- PKC-theta inhibitor 1
1160501-81-4
- $1820.00-3100.00
- TargetMol Chemicals Inc.
