ChemicalBook >> CAS DataBase List >>GI 254023X

GI 254023X

CAS No.
260264-93-5
Chemical Name:
GI 254023X
Synonyms
GI4023;GI 254023X;SRI 028594);GI 254023X(GI 4023;GI254023X[SML0789];GI254023X, 10 mM in DMSO;GI 254023X;GI-254023X;GI4023;SRI028594;GI254023X; GI 254023X; GI-254023X;GI4023; GI-4023; GI 4023;(R)-N-((S)-3,3-Dimethyl-1-(methylamino)-1-oxobutan-2-yl)-2-((S)-1-(N-hydroxyformamido)ethyl)-5-phenylpentanamide;(2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-2-[(1S)-1-(N-hydroxyformamido)ethyl]-5-phenylpentanamide
CBNumber:
CB82650737
Molecular Formula:
C21H33N3O4
Molecular Weight:
391.51
MDL Number:
MFCD19381832
MOL File:
260264-93-5.mol
MSDS File:
SDS
TDS File:
TDS
Last updated:2026-08-20 20:20:01
Product description Number Pack Size Price
GI254023X ≥98% (HPLC) SML0789 5mg $234
GI254023X ≥98% (HPLC) SML0789 25mg $933
GI 254023X ≥98% 28284 1mg $63
GI 254023X ≥98% 28284 5mg $183
GI 254023X ≥98% 28284 10mg $303

GI 254023X Properties

Density 1.112±0.06 g/cm3(Predicted)
storage temp. 2-8°C
solubility DMSO: soluble15mg/mL, clear
form powder
pka 8.48±0.69(Predicted)
color white to beige
InChIKey GHVMTHKJUAOZJP-CGTJXYLNSA-N
SMILES ON(C=O)[C@@H](C)[C@@H](CCCC1=CC=CC=C1)C(N[C@@H](C(C)(C)C)C(NC)=O)=O
UNSPSC Code 12352200
NACRES NA.77

SAFETY

Risk and Safety Statements

WGK Germany  3
Storage Class 11 - Combustible Solids

GI 254023X price More Price(56)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Sigma-Aldrich SML0789 GI254023X ≥98% (HPLC) 260264-93-5 5mg $234 2026-04-30 Buy
Sigma-Aldrich SML0789 GI254023X ≥98% (HPLC) 260264-93-5 25mg $933 2026-04-30 Buy
Cayman Chemical 28284 GI 254023X ≥98% 260264-93-5 1mg $63 2026-04-30 Buy
Cayman Chemical 28284 GI 254023X ≥98% 260264-93-5 5mg $183 2026-04-30 Buy
Cayman Chemical 28284 GI 254023X ≥98% 260264-93-5 10mg $303 2026-04-30 Buy
Product number Packaging Price Buy
SML0789 5mg $234 Buy
SML0789 25mg $933 Buy
28284 1mg $63 Buy
28284 5mg $183 Buy
28284 10mg $303 Buy

GI 254023X Chemical Properties,Uses,Production

Uses

GI 254023X is an ADAM10 metaloproteinase inhibitor.

Uses

GI254023X has been used to inhibit ADAM10 (ADAM metallopeptidase domain 10).

Definition

ChEBI: GI254023X is a L-valine derivative that is 3-methyl-L-valine in which carboxy OH group is replaced by a methylnitrilo group and the one of the amino hydrogens is replaced by a (2R)-2-{(1S)-1-[formyl(hydroxy)amino]ethyl}-5-phenylpentanoyl group. It is a potent MMP9 and ADAM10 metalloprotease inhibitor with IC50 of 2.5 and 5.3 nM, respectively. It has a role as an apoptosis inducer, an antineoplastic agent, a matrix metalloproteinase inhibitor and an EC 3.4.24.* (metalloendopeptidase) inhibitor. It is a L-valine derivative, an aldehyde and a member of hydroxylamines.

Biochem/physiol Actions

GI254023X is a potent and selective ADAM10 metalloproteinase inhibitor.

storage

Store at -20°C

GI 254023X Preparation Products And Raw materials

Raw materials

Preparation Products

GI 254023X Suppliers

Global( 140)Suppliers
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc.
+1-781-999-5354; +1-00000000000 marketing@targetmol.com United States 32431 58
Career Henan Chemica Co
+86-0371-86658258 +86-13203830695 laboratory@coreychem.com China 30203 58
TargetMol Chemicals Inc.
+1-781-999-5354; support@targetmol.com United States 38999 58
Zhengzhou Anbu Chem Co.,Ltd
+86-0371-88006763; +86-15988602810 sales@anbuchem.com China 3429 58
Aladdin Scientific
tp@aladdinsci.com United States 54746 58
Shaanxi Dideu New Materials Co. Ltd
18192503167 1036@dideu.com China 13233 58
NANJING YINGWEN BIOTECHNOLOGY CO LTD
+86-13382787392 sales@aeechem.com China 10002 58
Amadis Chemical Company Limited
571-89925085 sales@amadischem.com China 131885 58
Chembest Research Laboratories Limited 021-20908456 sales@BioChemBest.com China 5996 61
BOC Sciences 1-631-485-4226; 16314854226 info@bocsci.com United States 9920 65

View Lastest Price from GI 254023X manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
GI254023X pictures 2026-08-20 GI254023X
260264-93-5
$97.00-198.00 98.55% 10g TargetMol Chemicals Inc.
GI 254023X pictures 2026-06-30 GI 254023X
260264-93-5
1KG 98% 1000kg Shaanxi Dideu New Materials Co. Ltd
  • GI254023X pictures
  • GI254023X
    260264-93-5
  • $97.00-198.00
  • 98.55%
  • TargetMol Chemicals Inc.
  • GI 254023X pictures
  • GI 254023X
    260264-93-5
  • $0.00
  • 98%
  • Shaanxi Dideu New Materials Co. Ltd

GI 254023X Spectrum

GI 254023X (2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]-propyl]-2-[(1S)-1-[formyl(hydroxy)amino]ethyl]-5-phenylpentanamide GI4023 GI 254023X(GI 4023 SRI 028594) GI 254023X;GI-254023X;GI4023;SRI028594 (2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-2-[(1S)-1-(N-hydroxyformamido)ethyl]-5-phenylpentanamide ((2R,3S)-3-(formyl-hydroxyamino)-2-(3-phenyl-1-propyl)butanoic acid [(1S)-2,2-dimethyl-1-methylcarbamoyl-1-propyl] amide) (alphaR)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-alpha-[(1S)-1-(formylhydroxyamino)ethyl]benzenepentanamide GI254023X; GI 254023X; GI-254023X;GI4023; GI-4023; GI 4023 Benzenepentanamide, N-[(1S)-2,2-dimethyl-1-[(methylamino)carbonyl]propyl]-α-[(1S)-1-(formylhydroxyamino)ethyl]-, (αR)- (R)-N-((S)-3,3-Dimethyl-1-(methylamino)-1-oxobutan-2-yl)-2-((S)-1-(N-hydroxyformamido)ethyl)-5-phenylpentanamide GI254023X, 10 mM in DMSO GI254023X[SML0789] 260264-93-5 GI 254023X