GI 254023X
- CAS No.
- 260264-93-5
- Chemical Name:
- GI 254023X
- Synonyms
- GI4023;GI 254023X;SRI 028594);GI 254023X(GI 4023;GI254023X[SML0789];GI254023X, 10 mM in DMSO;GI 254023X;GI-254023X;GI4023;SRI028594;GI254023X; GI 254023X; GI-254023X;GI4023; GI-4023; GI 4023;(R)-N-((S)-3,3-Dimethyl-1-(methylamino)-1-oxobutan-2-yl)-2-((S)-1-(N-hydroxyformamido)ethyl)-5-phenylpentanamide;(2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-2-[(1S)-1-(N-hydroxyformamido)ethyl]-5-phenylpentanamide
- CBNumber:
- CB82650737
- Molecular Formula:
- C21H33N3O4
- Molecular Weight:
- 391.51
- MDL Number:
- MFCD19381832
- MOL File:
- 260264-93-5.mol
- MSDS File:
- SDS
- TDS File:
- TDS
| Product description | Number | Pack Size | Price |
| GI254023X ≥98% (HPLC) | SML0789 | 5mg | $234 |
| GI254023X ≥98% (HPLC) | SML0789 | 25mg | $933 |
| GI 254023X ≥98% | 28284 | 1mg | $63 |
| GI 254023X ≥98% | 28284 | 5mg | $183 |
| GI 254023X ≥98% | 28284 | 10mg | $303 |
| Density | 1.112±0.06 g/cm3(Predicted) |
|---|---|
| storage temp. | 2-8°C |
| solubility | DMSO: soluble15mg/mL, clear |
| form | powder |
| pka | 8.48±0.69(Predicted) |
| color | white to beige |
| InChIKey | GHVMTHKJUAOZJP-CGTJXYLNSA-N |
| SMILES | ON(C=O)[C@@H](C)[C@@H](CCCC1=CC=CC=C1)C(N[C@@H](C(C)(C)C)C(NC)=O)=O |
| UNSPSC Code | 12352200 |
| NACRES | NA.77 |
GI 254023X price More Price(56)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich | SML0789 | GI254023X ≥98% (HPLC) | 260264-93-5 | 5mg | $234 | 2026-04-30 | Buy |
| Sigma-Aldrich | SML0789 | GI254023X ≥98% (HPLC) | 260264-93-5 | 25mg | $933 | 2026-04-30 | Buy |
| Cayman Chemical | 28284 | GI 254023X ≥98% | 260264-93-5 | 1mg | $63 | 2026-04-30 | Buy |
| Cayman Chemical | 28284 | GI 254023X ≥98% | 260264-93-5 | 5mg | $183 | 2026-04-30 | Buy |
| Cayman Chemical | 28284 | GI 254023X ≥98% | 260264-93-5 | 10mg | $303 | 2026-04-30 | Buy |
GI 254023X Chemical Properties,Uses,Production
Uses
GI 254023X is an ADAM10 metaloproteinase inhibitor.
Uses
GI254023X has been used to inhibit ADAM10 (ADAM metallopeptidase domain 10).
Definition
ChEBI: GI254023X is a L-valine derivative that is 3-methyl-L-valine in which carboxy OH group is replaced by a methylnitrilo group and the one of the amino hydrogens is replaced by a (2R)-2-{(1S)-1-[formyl(hydroxy)amino]ethyl}-5-phenylpentanoyl group. It is a potent MMP9 and ADAM10 metalloprotease inhibitor with IC50 of 2.5 and 5.3 nM, respectively. It has a role as an apoptosis inducer, an antineoplastic agent, a matrix metalloproteinase inhibitor and an EC 3.4.24.* (metalloendopeptidase) inhibitor. It is a L-valine derivative, an aldehyde and a member of hydroxylamines.
Biochem/physiol Actions
GI254023X is a potent and selective ADAM10 metalloproteinase inhibitor.
storage
Store at -20°C
GI 254023X Preparation Products And Raw materials
Raw materials
Preparation Products
GI 254023X Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| TargetMol Chemicals Inc. | +1-781-999-5354; +1-00000000000 | marketing@targetmol.com | United States | 32431 | 58 |
| Career Henan Chemica Co | +86-0371-86658258 +86-13203830695 | laboratory@coreychem.com | China | 30203 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; | support@targetmol.com | United States | 38999 | 58 |
| Zhengzhou Anbu Chem Co.,Ltd | +86-0371-88006763; +86-15988602810 | sales@anbuchem.com | China | 3429 | 58 |
| Aladdin Scientific | tp@aladdinsci.com | United States | 54746 | 58 | |
| Shaanxi Dideu New Materials Co. Ltd | 18192503167 | 1036@dideu.com | China | 13233 | 58 |
| NANJING YINGWEN BIOTECHNOLOGY CO LTD | +86-13382787392 | sales@aeechem.com | China | 10002 | 58 |
| Amadis Chemical Company Limited | 571-89925085 | sales@amadischem.com | China | 131885 | 58 |
| Chembest Research Laboratories Limited | 021-20908456 | sales@BioChemBest.com | China | 5996 | 61 |
| BOC Sciences | 1-631-485-4226; 16314854226 | info@bocsci.com | United States | 9920 | 65 |
View Lastest Price from GI 254023X manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
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2026-08-20 | GI254023X
260264-93-5
|
$97.00-198.00 | 98.55% | 10g | TargetMol Chemicals Inc. | ||
![]() |
2026-06-30 | GI 254023X
260264-93-5
|
1KG | 98% | 1000kg | Shaanxi Dideu New Materials Co. Ltd |
-

- GI254023X
260264-93-5
- $97.00-198.00
- 98.55%
- TargetMol Chemicals Inc.
-

- GI 254023X
260264-93-5
- $0.00
- 98%
- Shaanxi Dideu New Materials Co. Ltd




