(R)-tert-butyl 4-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate

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(R)-tert-butyl 4-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate Basic information
Product Name:(R)-tert-butyl 4-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate
Synonyms:(R)-tert-butyl 4-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate;N-Boc-(R)-2-(3-Thiazolidinylcarbonyl)pyrrolidine;1-Pyrrolidinecarboxylic acid, 2-(3-thiazolidinylcarbonyl)-, 1,1-dimethylethyl ester, (R)- (9CI);(R)-tert-Butyl 2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate;(R)-2-(3-Thiazolidinylcarbonyl)-1-Pyrrolidinecarboxylic Acid 1,1-Dimethylethyl Ester
CAS:155251-72-2
MF:C13H22N2O3S
MW:286.39
EINECS:
Product Categories:
Mol File:155251-72-2.mol
(R)-tert-butyl 4-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate Structure
(R)-tert-butyl 4-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate Chemical Properties
Melting point 70-73°C
Boiling point 443.9±45.0 °C(Predicted)
density 1.226±0.06 g/cm3(Predicted)
storage temp. Refrigerator
solubility Chloroform (Slightly), Methanol (Slightly)
form Solid
pka-1.06±0.20(Predicted)
color Clear Colorless Thick Oil to White to Off-White
Safety Information
MSDS Information
(R)-tert-butyl 4-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate Usage And Synthesis
UsesN-Boc-(R)-2-(3-Thiazolidinylcarbonyl)-1-pyrrolidine, is an impurity of Teneligliptin (T018300), is a dipeptidyl peptidase-4 (DPP-4) inhibitor that is used to treat type 2 diabetes. It is eliminated via excretion, and has a half-life of 24.2 hours in the human body.
(R)-tert-butyl 4-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate Preparation Products And Raw materials
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