- Ocaperidone
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- $39.00 / 1mg
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2026-01-20
- CAS:129029-23-8
- Min. Order:
- Purity: 99.94%
- Supply Ability: 10g
- Ocaperidone USP/EP/BP
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- $1.10 / 1g
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2025-11-18
- CAS:129029-23-8
- Min. Order: 1g
- Purity: 99.9%
- Supply Ability: 100 Tons min
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| | Ocaperidone Basic information |
| Product Name: | Ocaperidone | | Synonyms: | Ocaperidone;Ocaperidona;3-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2,9-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one;3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2,9-dimethylpyrido[1,2-a]pyrimidin-4-one;R79598;4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2,9-dimethyl-;Ocaperidone USP/EP/BP;Ocaperidone (R79598) | | CAS: | 129029-23-8 | | MF: | C24H25FN4O2 | | MW: | 420.48 | | EINECS: | | | Product Categories: | | | Mol File: | 129029-23-8.mol |  |
| | Ocaperidone Chemical Properties |
| Melting point | 180.0 to 184.0 °C | | Boiling point | 588.0±60.0 °C(Predicted) | | density | 1.32 g/cm3 | | storage temp. | 2-8°C | | solubility | DMSO:16.0(Max Conc. mg/mL);38.1(Max Conc. mM) | | pka | 7.97±0.10(Predicted) | | form | powder to crystal | | color | White to Light yellow | | CAS DataBase Reference | 129029-23-8 |
| | Ocaperidone Usage And Synthesis |
| Uses | Antipsychotic. | | Definition | ChEBI: Ocaperidone is a pyridopyrimidine. | | in vivo | Ocaperidone shows a potent occupation of 5HT2 receptor via in vivo binding in the frontal cortex of rats with an ED50 of 0.04 mg/kg, and 0.1 4-0.1 6 mg/kg for D2 receptor in the striatum and the nucleus accumbens[1]. Ocaperidone (R 79598) antagonizes dopamine D2 and 5-HT2, and shows a a partial generalization to buspirone with an ED50 of 0.163 mg/kg[3]. | | IC 50 | 5-HT2 Receptor: 0.14 nM (Ki); a1-adrenergic receptor: 0.46 nM (Ki); D2 Receptor: 0.75 nM (Ki); Histamine H1: 1.6 nM (Ki); a2-adrenergic receptor: 5.4 nM (Ki); 5-HT1A Receptor: 7.6 (pEC50, h5-HT1A); 5-HT1A Receptor: 8.08 (pKi, h5-HT1A) |
| | Ocaperidone Preparation Products And Raw materials |
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