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2-METHYLINDOLE-3-ACETIC ACID

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Products Intro: Product Name:(2-Methyl-1H-indol-3-yl)acetic acid
CAS:1912-43-2
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CAS:1912-43-2
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CAS:1912-43-2
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Products Intro: Product Name:2-Methylindole-3-acetic acid
CAS:1912-43-2
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2-METHYLINDOLE-3-ACETIC ACID manufacturers

2-METHYLINDOLE-3-ACETIC ACID Basic information
Product Name:2-METHYLINDOLE-3-ACETIC ACID
Synonyms:(2-METHYL-1H-INDOL-3-YL)-ACETIC ACID;2-METHYL-3-INDOLEACETIC ACID;2-METHYLINDOLE-3-ACETIC ACID;AKOS BC-0002;IFLAB-BB F0345-1687;2-Me-IAA;2-METHYLINDOLE-3-ACETIC ACID(2MeIAA);2-Methyl Indole-3-acetate Acid
CAS:1912-43-2
MF:C11H11NO2
MW:189.21
EINECS:000-000-0
Product Categories:Imidazol&Benzimidazole;Indoles and derivatives;Building Blocks;Heterocyclic Building Blocks;Indoles
Mol File:1912-43-2.mol
2-METHYLINDOLE-3-ACETIC ACID Structure
2-METHYLINDOLE-3-ACETIC ACID Chemical Properties
Melting point 205 °C (dec.) (lit.)
Boiling point 418.2±30.0 °C(Predicted)
density 1.299±0.06 g/cm3(Predicted)
storage temp. 2-8°C(protect from light)
solubility DMSO (Slightly), Methanol (Slightly)
form Solid
pka4.19±0.30(Predicted)
color Pale Brown to Light Brown
BRN 152701
InChI1S/C11H11NO2/c1-7-9(6-11(13)14)8-4-2-3-5-10(8)12-7/h2-5,12H,6H2,1H3,(H,13,14)
InChIKeyQJNNHJVSQUUHHE-UHFFFAOYSA-N
SMILESCc1[nH]c2ccccc2c1CC(O)=O
CAS DataBase Reference1912-43-2(CAS DataBase Reference)
Safety Information
Hazard Codes Xi
Safety Statements 22-24/25
WGK Germany 3
HazardClass IRRITANT
Storage Class11 - Combustible Solids
MSDS Information
ProviderLanguage
SigmaAldrich English
ALFA English
2-METHYLINDOLE-3-ACETIC ACID Usage And Synthesis
Uses2-Methylindole-3-acetic Acid is a derivative of Indole-3-acetic acid which is a plant growth regulator. It induces cell division and cell elongation that promotes plant growth.
DefinitionChEBI: 2-Methylindole-3-acetic acid is a member of indole-3-acetic acids.
General Description2-Methyl-3-indoleacetic acid is a common plant growth hormone. Relative activity of 2-methyl-3-indoleacetic acid in promoting growth (elongation) in plant cells was evaluated.
Synthesis
Levulinic acid

123-76-2

Phenylhydrazine

100-63-0

2-METHYLINDOLE-3-ACETIC ACID

1912-43-2

GENERAL METHOD: Acetylpropionic acid (10 mmol) was dissolved in acetic acid (30 mL) and phenylhydrazine (15 mmol) was added to the solution under stirring conditions. The reaction mixture was heated to reflux for 4 hours. Upon completion of the reaction, it was cooled to room temperature and the mixture was poured into water (200 mL) and the pH was adjusted to 5-6 with 30% sodium hydroxide solution.The precipitated solid was collected by filtration, recrystallized from ethanol and dried under vacuum to give 2-methylindole-3-acetic acid (2a). 2-Methylindole-3-acetic acid (2a): yellow solid, 78% yield, melting point 200-203 °C (literature value 199-200 °C); 1H NMR (500 MHz, CDCl3) δ: 2.31 (3H, s, CH3), 3.65 (2H, s, CH2), 6.97 (1H, t, J = 7.5 Hz, ArH), 7.12 ( 1H, t, J = 7.5 Hz, ArH), 7.23 (1H, d, J = 6.0 Hz, ArH), 7.33 (1H, d, J = 6.0 Hz, ArH), 10.83 (1H, s, COOH), 12.15 (1H, s, NH); IR (νmax, cm-1): 1504, 1518, 1565, 1624, 1769, 2935, 3001, 3535; HRMS m/z: 190.0824 (calculated value C11H11NO2 [M + H]+: 190.0823).

References[1] Journal of Chemical Research, 2016, vol. 40, # 10, p. 588 - 590
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