| Company Name: |
Tianjin Kailiqi Biotechnology Co., Ltd.
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| Tel: |
15076683720 |
| Email: |
klq@cw-bio.com |
| Products Intro: |
Product Name:CB1R Allosteric modulator 3
CAS:2633686-36-7
Purity:大于98% Package:1g,5g,10g,25g根据客户需要分装 Remarks:Not For Human Use, Lab Use Only.
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| Company Name: |
Shanghai Yifei Biotechnology Co. , Ltd.
|
| Tel: |
021-65675885 18964387627 |
| Email: |
customer_service@efebio.com |
| Products Intro: |
Product Name:CB1R Allosteric modulator 3
CAS:2633686-36-7
Purity:98% Package:1mg;5mg;10mg
|
| Company Name: |
TargetMol Chemicals Inc.
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| Tel: |
15002134094 |
| Email: |
marketing@targetmol.cn |
| Products Intro: |
Product Name:CB1R Allosteric modulator 3
CAS:2633686-36-7
Purity:98.18% Package:1mg/RMB 347;5mg/RMB 828;10mg/RMB 1380
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1H-Indole, 3-[1-(2-chlorophenyl)-2-nitroethyl]-2-phenyl- manufacturers
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| | 1H-Indole, 3-[1-(2-chlorophenyl)-2-nitroethyl]-2-phenyl- Basic information |
| | 1H-Indole, 3-[1-(2-chlorophenyl)-2-nitroethyl]-2-phenyl- Chemical Properties |
| Boiling point | 604.7±55.0 °C(Predicted) | | density | 1.306±0.06 g/cm3(Predicted) | | pka | 7.57±0.18(Predicted) | | form | Solid | | color | Off-white to light yellow |
| | 1H-Indole, 3-[1-(2-chlorophenyl)-2-nitroethyl]-2-phenyl- Usage And Synthesis |
| Uses | CB1R Allosteric modulator 3 is a CB1R positive allosteric modulator. CB1R Allosteric modulator 3 has potent inhibition of cAMP and β-Arrestin with EC50 values of 0.018 μM and 1.241 μM, respectively[1]. | | IC 50 | CB1 | | References | [1] Peter C Schaffer, et al. Focused structure-activity relationship profiling around the 2-phenylindole scaffold of a cannabinoid type-1 receptor agonist-positive allosteric modulator: site-III aromatic-ring congeners with enhanced activity and solubility. Bioorg Med Chem. 2020 Nov 1;28(21):115727. DOI:10.1016/j.bmc.2020.115727 |
| | 1H-Indole, 3-[1-(2-chlorophenyl)-2-nitroethyl]-2-phenyl- Preparation Products And Raw materials |
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