| Company Name: |
SPIRO PHARMA |
| Tel: |
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| Email: |
eric_feng1954@126.com |
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| | Sumanirole maleate Basic information |
| Product Name: | Sumanirole maleate | | Synonyms: | (5R)-5,6-Dihydro-5-(MethylaMino)-4H-iMidazo[4,5,1-ij]quinolin-2(1H)-one (2Z)-2-Butenedioate;(R)-5,6-Dihydro-5-(MethylaMino)-4H-iMidazo[4,5,1-ij]quinolin-
2(1H)-one (2Z)-2-Butenedioate;(R)-5-(MethylaMino)-5,6-dihydro-1H-iMidazo[4,5,1-ij]quinolin-2(4H)-one Maleate,(free base);4H-IMidazo[4,5,1-ij]quinolin-2(1H)-one,5,6-dihydro-5-(MethylaMino)-, (5R)-;(5R)-5,6-Dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one;Sumanirole | | CAS: | 179386-43-7 | | MF: | C11H13N3O | | MW: | 203.24 | | EINECS: | | | Product Categories: | | | Mol File: | 179386-43-7.mol |  |
| | Sumanirole maleate Chemical Properties |
| density | 1.32 | | storage temp. | 2-8°C(protect from light) |
| | Sumanirole maleate Usage And Synthesis |
| Chemical Properties | Off-White to Light Beige Solid | | Uses | Sumanirole is a high affinity D2 receptor agonist (EC50 values are between 17 and 75 nM in cell-based assays). Sumanirole displays >200-fold selectivity for the D2 receptor against other dopamine rece
ptor subtypes (Ki values are 9.0, 1940, >2190 and >7140 for D2, D3, D4 and D1 receptors respectively). Sumanirole exhibits antiParkinsonian activity similar to Ropinirole (R641000). | | IC 50 | D2 Receptor |
| | Sumanirole maleate Preparation Products And Raw materials |
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