BCN-exo-PEG3-maleimide?Chemical Structure

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BCN-exo-PEG3-maleimide?Chemical Structure Basic information
Product Name:BCN-exo-PEG3-maleimide?Chemical Structure
Synonyms:BCN-exo-PEG3-maleimide?Chemical Structure;5,8,11-Trioxa-2,14-diazaheptadecanoic acid, 17-(2,5-dihydro-2,5-dioxo-1H-pyrrol-1-yl)-15-oxo-, (1α,8α,9α)-bicyclo[6.1.0]non-4-yn-9-ylmethyl ester;exo-BCN-PEG3-NHCO-Maleimide
CAS:2919127-00-5
MF:C26H37N3O8
MW:519.59
EINECS:
Product Categories:PEG
Mol File:2919127-00-5.mol
BCN-exo-PEG3-maleimide?Chemical Structure Structure
BCN-exo-PEG3-maleimide?Chemical Structure Chemical Properties
Boiling point 734.529±60.00 °C(Press: 760.00 Torr)(predicted)
density 1.269±0.10 g/cm3(Temp: 25 °C; Press: 760 Torr)(predicted)
pka12.050±0.46(predicted)
Safety Information
MSDS Information
BCN-exo-PEG3-maleimide?Chemical Structure Usage And Synthesis
UsesBCN-exo-PEG3-maleimide is an ADC Linker containing 3 PEG units. BCN-exo-PEG3-maleimide contains the lyophilic bidentate macrocyclic ligand BCN, which enables the further synthesis of macrocyclic complexes. In click chemistry, BCN reacts with molecules containing azide groups to form stable triazoles in the absence of catalysts. Its maleimide group (-Maleimide) degrades in aqueous media and has been used in drug delivery studies.
BCN-exo-PEG3-maleimide?Chemical Structure Preparation Products And Raw materials
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(R)-TCO4-PEG2-Maleimide Mal-amido-PEG9-NHBoc TCO4-PEG7-Maleimide SCO-PEG7-Maleimide BCN-exo-PEG2-Maleimide 5,8,11,14,17,20,23-Heptaoxa-2,26-diazanonacosanoic acid, 29-(2,5-dihydro-2,5-dioxo-1H-pyrrol-1-yl)-27-oxo-, (1R,8S)-bicyclo[6.1.0]non-4-yn-9-ylmethyl ester, rel-