PKG Inhibitor (trifluoroacetate salt)

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PKG Inhibitor (trifluoroacetate salt) Suppliers list
Company Name: Cayman Chemical Company  
Tel: 800-364-9897
Email: sales@caymanchem.com
PKG Inhibitor (trifluoroacetate salt) Basic information
Product Name:PKG Inhibitor (trifluoroacetate salt)
Synonyms:PKG Inhibitor (trifluoroacetate salt)
CAS:
MF:
MW:0
EINECS:
Product Categories:
Mol File:Mol File
PKG Inhibitor (trifluoroacetate salt) Structure
PKG Inhibitor (trifluoroacetate salt) Chemical Properties
solubility DMF: 5 mg/ml
DMSO: 15 mg/mlPBS (pH 7.2): 10 mg/ml
Safety Information
MSDS Information
PKG Inhibitor (trifluoroacetate salt) Usage And Synthesis
DescriptionPKG inhibitor is a specific cGMP-dependent PKG inhibitor (Ki = 86 µM).1 This synthetic peptide is a nonphosphorylatable analog of a substrate corresponding to the serine-32 phosphorylation site in histone H2B.1 PKG inhibitor has been reported to block cGMP-dependent NMDA potentiation and nitric oxide-induced depression of GABA currents in cultured retinal amacrine cells.2WARNING This product is not for human or veterinary use.
References[1] GLASS D B. Differential responses of cyclic GMP-dependent and cyclic AMP-dependent protein kinases to synthetic peptide inhibitors.[J]. Biochemical Journal, 1983, 213 1: 159-164. DOI: 10.1042/bj2130159
[2] E M WEXLER  S N  P K Stanton. Nitric oxide depresses GABAA receptor function via coactivation of cGMP-dependent kinase and phosphodiesterase.[J]. Journal of Neuroscience, 1998, 18 7: 2342-2349.
PKG Inhibitor (trifluoroacetate salt) Preparation Products And Raw materials
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