MT-802 manufacturers
- MT-802
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- $0.00 / 1mg
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2026-01-04
- CAS:2231744-29-7
- Min. Order: 1mg
- Purity: 98%min
- Supply Ability: 50mg
- MT-802
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- $88.00 / 1mg
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2025-12-25
- CAS:2231744-29-7
- Min. Order:
- Purity: 97.00%
- Supply Ability: 10g
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| Product Name: | MT-802 | | Synonyms: | MT-802;Acetamide, 2-[2-[2-[4-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]-1-piperidinyl]ethoxy]ethoxy]-N-[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-5-yl]-;2-[2-[2-[4-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]-1-piperidinyl]ethoxy]ethoxy]-N-[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-5-yl]-;2-(2-(2-(4-(4-Amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)ethoxy)ethoxy)-N-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)acetamide;MT802,inhibit,Inhibitor,Btk,Bruton tyrosine kinase,MT-802,MT 802,PROTACs;MT-802, 10 mM in DMSO | | CAS: | 2231744-29-7 | | MF: | C41H41N9O8 | | MW: | 787.82 | | EINECS: | | | Product Categories: | | | Mol File: | 2231744-29-7.mol |  |
| | MT-802 Chemical Properties |
| storage temp. | Store at -20°C | | solubility | DMSO: 100 mg/mL (126.93 mM) | | form | Solid | | color | White to off-white |
| | MT-802 Usage And Synthesis |
| Uses | MT-802 is a potent BTK degrader based on Cereblon ligand, with a DC50 of 1 nM. MT-802 has potential to treat C481S mutant chronic lymphocytic leukemia (CLL)[1]. | | References | [1] Buhimschi AD, et al. Targeting the C481S Ibrutinib-Resistance Mutation in Bruton's Tyrosine Kinase Using PROTAC-Mediated Degradation. Biochemistry. 2018 Jul 3;57(26):3564-3575. DOI:10.1021/acs.biochem.8b00391 |
| | MT-802 Preparation Products And Raw materials |
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