- Antide acetate
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- $196.00 / 1mg
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2026-01-04
- CAS:
- Min. Order:
- Purity: 99.57%
- Supply Ability: 10g
- Antide
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- $70.00 / 1kg
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2025-06-03
- CAS:112568-12-4
- Min. Order: 10kg
- Purity: 0.99
- Supply Ability: 20tons
- Antide
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- $0.00 / 1kg
-
2025-04-04
- CAS:112568-12-4
- Min. Order: 1kg
- Purity: 98%
- Supply Ability: 1Ton
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| Product Name: | Antide | | Synonyms: | iturelix;Ac-D-2-Nal-4-chloro-D-Phe-beta-(3-pyridyl)-D-Ala-Ser-Lys(nicotinoyl)-D-Lys(nicotinoyl)-Leu-Lys(isopropyl)-Pro-D-Ala-NH2;AC-DNAL-D: P-CLPHE-DPAL-SER-LYS: NICOTINOYL-DLYS: NICOTINOYL-LEU-LYS: ISOPROPYL-PRO-DALA-NH2;Brn 4866881;D-Alaninamide, N-acetyl-3-(2-naphthalenyl)-D-alanyl-4-chloro-D-phenylalanyl-3-(3-pyridinyl)-D-alanyl-L-seryl-N(sup 6)-(3-pyridinylcarbonyl)-L-lysyl-N(sup 6)-(3-pyridinylcarbonyl)-D-lysyl-L-leucyl-N(sup 6)-(1-methylethyl)-L-lysyl-L-prolyl-;D-Alaninamide, N-acetyl-3-(2-naphthalenyl)-D-alanyl-4-chloro-D-phenylalanyl-3-(3-pyridinyl)-D-alanyl-L-seryl-N6-(3-pyridinylcarbonyl)-L-lysyl-N6-(3-pyridinylcarbonyl)-D-lysyl-L-leucyl-N6-(1-methylethyl)-L-lysyl-L-prolyl-;Orf 23541;Ac-D-2-Nal-4-chloro-D-Phe-b-(3-pyridyl)-D-Ala-Ser-Lys(nicotinoyl)-D-Lys(nicotinoyl)-Leu-Lys(isopropyl)-Pro-D-Ala-NH2 | | CAS: | 112568-12-4 | | MF: | C82H108ClN17O14 | | MW: | 1591.29 | | EINECS: | | | Product Categories: | hormones;Peptide;LH-RH;LH-RHPeptides for Cell Biology;Neuropeptides;Releasing Factors | | Mol File: | 112568-12-4.mol |  |
| | Antide Chemical Properties |
| Boiling point | 1798.0±65.0 °C(Predicted) | | density | 1.258±0.06 g/cm3(Predicted) | | storage temp. | −20°C | | form | Solid | | pka | 12.78±0.46(Predicted) | | color | White to off-white | | InChIKey | QRYFGTULTGLGHU-NBERXCRTSA-N |
| Hazard Codes | T | | Risk Statements | 60 | | Safety Statements | 53-22-36/37/39-45 | | WGK Germany | 3 | | RTECS | AY2961700 | | HS Code | 3504009000 |
| | Antide Usage And Synthesis |
| Uses | Reversible inhibition of gonadotropin secretion and subsequent suppression of ovarian and testicular steroid secretio (gonadotropin releasing hormone antagonist). | | Uses | Antide, is a GnRH and LH-RH antagonist, and with high anti-ovulatory and negligible histamine release activity. | | in vivo | Antide (subcutaneously; 1, 3, 6, 10 and 15 mg/kg; once or on 5 consecutive days) can induce a long-term chemical castration in adult male rats and cynomolgus monkeys[1]. | Animal Model: | Cynomolgus monkey and rat[1] | | Dosage: | 1, 3, 6, 10 and 15 mg/kg | | Administration: | Subcutaneous, once or on 5 consecutive days | | Result: | Had a dose-dependent inhibitory effect on serum concentration of LH (only rat) and testosterone and on the weights of the testes, prostates and seminal vesicles.
Achieved long-lasting castration-like effects at concentrations between 6 (less than or equal to 8 weeks) and 15 mg/kg (greater than 8 weeks) in the rat.
Induced a prolonged inhibitory effect only at 15 mg/kg and the duration was only 2-3 weeks in the cynomolgus monkey.
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| | Description | Antide acetate (Ac-AA10-NH2) is an LHRH antagonist and represses LH and FSH release from the pituitary gland. Antide Mw is 1590.6 Dalton. |
| | Antide Preparation Products And Raw materials |
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