| Company Name: |
TargetMol Chemicals Inc.
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| Tel: |
15002134094 |
| Email: |
marketing@targetmol.cn |
| Products Intro: |
Product Name:TP-680
CAS:176915-07-4
Package:25mg/RMB 10600;50mg/RMB 13800;100mg/RMB 17500
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3-Pyridinecarboxylic acid, 2-[[(2R)-3-[4-(diphenylmethyl)-1-piperazinyl]-2-[(1H-indol-2-ylcarbonyl)amino]-3-oxopropyl]thio]- (9CI) manufacturers
- TP-680
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- $1520.00 / 25mg
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2025-08-21
- CAS:176915-07-4
- Min. Order:
- Purity:
- Supply Ability: 10g
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| | 3-Pyridinecarboxylic acid, 2-[[(2R)-3-[4-(diphenylmethyl)-1-piperazinyl]-2-[(1H-indol-2-ylcarbonyl)amino]-3-oxopropyl]thio]- (9CI) Basic information |
| | 3-Pyridinecarboxylic acid, 2-[[(2R)-3-[4-(diphenylmethyl)-1-piperazinyl]-2-[(1H-indol-2-ylcarbonyl)amino]-3-oxopropyl]thio]- (9CI) Chemical Properties |
| Boiling point | 889.3±65.0 °C(Predicted) | | density | 1.40±0.1 g/cm3(Predicted) | | pka | 2.79±0.36(Predicted) |
| | 3-Pyridinecarboxylic acid, 2-[[(2R)-3-[4-(diphenylmethyl)-1-piperazinyl]-2-[(1H-indol-2-ylcarbonyl)amino]-3-oxopropyl]thio]- (9CI) Usage And Synthesis |
| Description | TP-680 is a new cholecystokininA receptor antagonist. | | Uses | TP-680 is a cholecystokinin receptor antagonist. TP-680 binds 1510 times more strongly to rat pancreatic CCKA receptors (IC50=1.2 nM) than to rat brain CCKB receptors (IC50=1812.5 nM). TP-680 can be used in the study of gastrointestinal diseases[1]. | | IC 50 | CCKAR: 1.2 nM (IC50); CCKBR: 1812.5 nM (IC50) | | References | [1] Akiyama T, et al. Pharmacological profile of TP-680, a new cholecystokininA receptor antagonist[J]. British journal of pharmacology, 1996, 117(7): 1558. DOI:10.1111/j.1476-5381.1996.tb15321.x |
| | 3-Pyridinecarboxylic acid, 2-[[(2R)-3-[4-(diphenylmethyl)-1-piperazinyl]-2-[(1H-indol-2-ylcarbonyl)amino]-3-oxopropyl]thio]- (9CI) Preparation Products And Raw materials |
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