Kinase inhibitor-1

Kinase inhibitor-1 Suppliers list
Company Name: TargetMol Chemicals Inc.
Tel: +1-781-999-5354; +17819995354
Email: marketing@targetmol.com
Products Intro: Product Name:Tarlox-TKI
CAS:2135696-72-7
Purity:97.03% Package:1mg;148USD Remarks:REAGENT;FOR LABORATORY USE ONLY
Company Name: TargetMol Chemicals Inc.
Tel: +1-781-999-5354;
Email: support@targetmol.com
Products Intro: Product Name:Tarlox-TKI
CAS:2135696-72-7
Purity:97.03% Package:1mg;148USD
Company Name: Wuhan Jingkang en Biomedical Technology Co., Ltd
Tel: +8613720134139
Email: orders@jknbiochem.com
Products Intro: Product Name:Kinase inhibitor 1
CAS:2135696-72-7
Purity:0.98 Package:10G:100G
Company Name: Shanghai EFE Biological Technology Co., Ltd.  
Tel: 021-65675885 18964387627
Email: info@efebio.com
Products Intro: Product Name:Tarlox-TKI
CAS:2135696-72-7
Purity:97.00% Package:1mg
Company Name: Shanghai YuanYe Biotechnology Co., Ltd.  
Tel: 021-61312847; 18021002903
Email: 3008007409@qq.com
Products Intro: Product Name:Tarlox-TKI
CAS:2135696-72-7
Package:1ml Remarks:T97014

Kinase inhibitor-1 manufacturers

  • Tarlox-TKI
  • Tarlox-TKI pictures
  • $148.00 / 1mg
  • 2026-04-22
  • CAS:2135696-72-7
  • Min. Order:
  • Purity: 97.03%
  • Supply Ability: 10g
  • Tarlox-TKI
  • Tarlox-TKI pictures
  • $148.00 / 1mg
  • 2026-04-22
  • CAS:2135696-72-7
  • Min. Order:
  • Purity: 97.03%
  • Supply Ability: 10g
Kinase inhibitor-1 Basic information
Product Name:Kinase inhibitor-1
Synonyms:Kinase inhibitor-1;2-Butenamide, N-[4-[(3-bromo-4-chlorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-4-(dimethylamino)-, (2E)-;Tarlox-TKI;TarloxTKI,Tarlox TKI
CAS:2135696-72-7
MF:C19H18BrClN6O
MW:461.74
EINECS:
Product Categories:
Mol File:2135696-72-7.mol
Kinase inhibitor-1 Structure
Kinase inhibitor-1 Chemical Properties
Boiling point 647.4±55.0 °C(Predicted)
density 1.552±0.06 g/cm3(Predicted)
storage temp. Store at -20°C
solubility DMSO: 100 mg/mL (216.57 mM); Water: < 0.1 mg/mL (insoluble)
form Solid
pka9.68±0.43(Predicted)
color Light yellow to yellow
Safety Information
MSDS Information
Kinase inhibitor-1 Usage And Synthesis
UsesTarlox-TKI, the active metabolite of Tarloxotinib, is an irreversible pan-ErbB TKI (Tarlox-TKI)[1].
IC 50EGFR
References[1] Victoria Jackson-Patel, et al. Hypoxia tumour targeting with Tarloxotinib to improve clinical outcomes for patients with EGFR-dependent malignancies.
Kinase inhibitor-1 Preparation Products And Raw materials
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