N-[4-Methyl-9-(1-methylethyl)-9H-carbazol-3-yl]-4-morpholinecarboxamide manufacturers
- NPY 5RA972
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2026-07-01
- CAS:439861-56-0
- Min. Order: 1KG
- Purity: 98%
- Supply Ability: 20Tons
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| | N-[4-Methyl-9-(1-methylethyl)-9H-carbazol-3-yl]-4-morpholinecarboxamide Basic information |
| | N-[4-Methyl-9-(1-methylethyl)-9H-carbazol-3-yl]-4-morpholinecarboxamide Chemical Properties |
| storage temp. | Store at RT | | solubility | Soluble to 100 mM in DMSO | | form | Powder | | color | White to off-white |
| | N-[4-Methyl-9-(1-methylethyl)-9H-carbazol-3-yl]-4-morpholinecarboxamide Usage And Synthesis |
| Uses | NPY 5RA972 is a potent antagonist of the neuropeptide Y5 receptor. | | in vivo | NPY5RA-972(p.o., 10.5 mg/kg) has a Tmax value of 1 hour in rats, a Cmax of 35 μM, a half-life of 6.4 hours, and a total plasma concentration of greater than 3 μM/h even 24 hours after administration[1].
NPY5RA-972 (p.o., 1-10 mg/kg) inhibits food intake elicited by a selective NPY Y5 receptor agonist, but has no effect on food intake or body weight in freely-fed Wistar rats or diet-obese rats Influence[1].
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| | N-[4-Methyl-9-(1-methylethyl)-9H-carbazol-3-yl]-4-morpholinecarboxamide Preparation Products And Raw materials |
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