3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)-

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3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)- Suppliers list
Company Name: ATK CHEMICAL COMPANY LIMITED
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Email: ivan@atkchemical.com
Products Intro: Product Name:GSK251
CAS:2125968-05-8
Purity:98% Package:10MG;50MG;100MG,1G,5G,10G.100G
Company Name: TargetMol Chemicals Inc.
Tel: +1-781-999-5354; +17819995354
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Products Intro: Product Name:GSK251
CAS:2125968-05-8
Purity:98.9% Package:1mg;166USD|5mg;417USD|10mg;592USD
Company Name: ShenZhen Trendseen Biological Technology Co.,Ltd.
Tel: 13417589054
Email: trendseenbio@gmail.com
Products Intro: Product Name:N-（2-（2-fluoro-4-（（4-isopropylpiperazin-1-yl）methyl）phenyl）pyridin-4-yl）-2-methoxy-5-morpholinopyridine-3-sulfonamide
CAS:2125968-05-8
Purity:99% Package:1kg；25kg
Company Name: Wuhan Jingkang en Biomedical Technology Co., Ltd
Tel: +8613720134139
Email: orders@jknbiochem.com
Products Intro: Product Name:GSK251
CAS:2125968-05-8
Purity:0.98 Package:10G:100G
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Products Intro: CAS:2125968-05-8
Purity:98%

3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)- manufacturers

  • GSK251
  • GSK251 pictures
  • $166.00 / 1mg
  • 2026-04-17
  • CAS:2125968-05-8
  • Min. Order:
  • Purity: 99.80%
  • Supply Ability: 10g
3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)- Basic information
Product Name:3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)-
Synonyms:3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)-;GSK251;N-（2-（2-fluoro-4-（（4-isopropylpiperazin-1-yl）methyl）phenyl）pyridin-4-yl）-2-methoxy-5-morpholinopyridine-3-sulfonamide;GSK251,GSK-251;N-[2-(2-fluoro-4-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)pyridin-4-yl]-2-methoxy-5-(morpholin-4-yl)pyridine-3-sulfonamide
CAS:2125968-05-8
MF:C29H37FN6O4S
MW:584.71
EINECS:
Product Categories:
Mol File:2125968-05-8.mol
3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)- Structure
3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)- Chemical Properties
Boiling point 742.4±70.0 °C(Predicted)
density 1.295±0.06 g/cm3(Predicted)
storage temp. Store at -20°C
solubility DMSO : 62.5 mg/mL (106.89 mM; ultrasonic and warming and heat to 60°C)
form Solid
pka-0.07±0.10(Predicted)
color Off-white to light yellow
Safety Information
MSDS Information
3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)- Usage And Synthesis
UsesGSK251 is a highly potent, highly selective, orally bioavailable inhibitor of PI3Kδ with a novel binding mode.
References[1] Down K, et al. Discovery of GSK251: A Highly Potent, Highly Selective, Orally Bioavailable Inhibitor of PI3Kδ with a Novel Binding Mode. J Med Chem. 2021 Sep 23;64(18):13780-13792. DOI:10.1021/acs.jmedchem.1c01102
3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)- Preparation Products And Raw materials
Tag:3-Pyridinesulfonamide, N-[2-[2-fluoro-4-[[4-(1-methylethyl)-1-piperazinyl]methyl]phenyl]-4-pyridinyl]-2-methoxy-5-(4-morpholinyl)-(2125968-05-8) Related Product Information