Anamorelin Fumarate NEW
| Price | $1670 | $2180 | $2800 |
| Package | 25mg | 50mg | 100mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-10-27 |
Product Details
| Product Name: Anamorelin Fumarate | CAS No.: 339539-92-3 |
| Supply Ability: 10g | Release date: 2025/10/27 |
Product Introduction
Bioactivity
| Name | Anamorelin Fumarate |
| Description | Anamorelin Fumarate is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay). |
| In vitro | No significant antagonist activity is observed with Anamorelin at concentrations of up to 1,000 nM. In the binding experiments, Anamorelin binds to the ghrelin receptor with a binding affinity constant (Ki) of 0.70 nM. In the competition assay with radiolabeled ibutamoren (another ghrelin receptor agonist), Anamorelin is also found to bind with high affinity to the ghrelin receptor (IC50: 0.69 nM). In rat pituitary cells incubated with Anamorelin, there is a dose-dependent stimulatory effect on GH release and the potency (EC50) is 1.5 nM. Anamorelin is screened for activity against a set of over 100 receptors, ion channels, transporters, and enzymes. Anamorelin demonstrates binding to the tachykinin neurokinin 2 (NK2) site (IC50: 0.021 μM); however, a subsequent NK2 functional assay demonstrates no functional activity. |
| In vivo | In rats, oral administration of Anamorelin at doses of 3, 10, or 30 mg/kg once daily significantly enhanced food intake and body weight from Day 2 to Day 7 of treatment, compared to the vehicle control. The observed increases in food consumption and weight gain were dose-dependent and statistically significant across all dosage levels when compared to the control group. Additionally, a single oral dose of Anamorelin at 3, 10, or 30 mg/kg resulted in a dose-dependent elevation in plasma GH levels and GH AUC0-6h. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Keywords | RC-1291 Fumarate | RC 1291 Fumarate | ONO7643 Fumarate | ONO 7643 Fumarate | ghrelin receptor | Anamorelin Fumarate |
| Inhibitors Related | Ibutamoren Mesylate | YIL 781 | AnaMorelin hydrochloride | Capromorelin Tartrate | Anamorelin | Ibutamoren | CJC-1295 acetate(863288-34-0 free base) | L-692429 | TC-G-1008 | Human growth hormone-releasing factor acetate | TM-N1324 | Cortistatin-8 acetate |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries， 10000+ Noval Small Molecucles，16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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