英文名称:PSMA I&T
DOTAGA-DTyr(3I)-DPhe-DLys(Sub-Lys-urea-Glu)
CAS NO:2192281-54-0
序列号:DOTAGA-DTyr(3I)-DPhe-DLys(Sub-Lys-urea-Glu)
IUPAC Name:(2S)-2-[[(1S)-1-carboxy-5-[[8-[[(5R)-5-carboxy-5-[[(2R)-2-[[(2R)-2-[[4-carboxy-4-[4,7,10-tris(carboxymethyl)-1,4,7,10-tetrazacyclododec-1-yl]butanoyl]amino]-3-(4-hydroxy-3-iodophenyl)propanoyl]amino]-3-phenylpropanoyl]amino]pentyl]amino]-8-oxooctanoyl]amino]pentyl]carbamoylamino]pentanedioic acid
分子式:C63H92IN11O23
分子量:1498.3
存储温度:2-8℃
纯度:≥95%
溶解性:溶于二甲基亚砜
结构式:

177 Lu-PSMA-I&T是放射性标记肽。PSMA I&T也标记有68 Ga和111 In,分别用于PET和SPECT成像(也包括无线电引导手术)。
其他PSMA系列试剂:
PSMA617 1702967-37-0
PSMA11 1366302-52-4
PSMA1007 2093321-19-6
HYNIC-PSMA
DCL (PSMA inhibitor) (ACUPA)
NOTA-PSMA 1575386-67-2
tert-Butyl-DCL (PSMA inhibitor) 1025796-31-9
PSMA-ligand-1 1610413-97-2
PSMA-BCH
PSMA I&T
PSMA I&F
关键字: 2192281-54-0;PSMA I&T;双功能螯合剂;