中文名:宁格替尼
英文名:Ningetinib
纯度:Moligand™,≥98%
货号:N413663
Cas号:1394820-69-9
存储温度:-20°C储存
运输条件:超低温运输
产品介绍:
Information
Ningetinib (CT-053, DE-120, CT053PTSA) is a potent, orally bioavailable inhibitor oftyrosine kinasewith IC50 of 6.7 nM, 1.9 nM and <1.0 nM forc-Met,VEGFR2andAxl, respectively. Ningetinib exhibits antitumor activity.
Targets
Axl (Cell-free assay); VEGFR2 (Cell-free assay); c-Met (Cell-free assay) 1.0 nM; 1.9 nM; 6.7 nM
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