中文名:喹吖因 二盐酸盐
英文名:Quinacrine dihydrochloride
纯度:≥98%
货号:Q113496
Cas号:69-05-6
存储温度:避光
运输条件:常规运输
产品介绍:
Quinacrine dihydrochloride is a non-specific PLA2 (phospholipase A2) inhibitor. Quinacrine, Dihydrochloride acts as an AChR (acetylcholine receptor) antagonist. Quinacrine dihydrochloride suppresses glibenclamide-sensitive K+-currents (IC50 = 4.4 μM). This compound also inhibits MAO (monoamine oxidase). Quinacrine, Dihydrochloride is an inhibitor of cPLA2, MAO-A and MAO-B.
A non-specific PLA2 inhibitor. and acetylcholine receptor antagonist
Application:
Quinacrine dihydrochloride has been used:
in its uptake and accumulation studies in mouse lung slices using fluorescence microscope
in the staining of ATP vesicles in mesenchymal stem cells (MSCs)
in uptake-release assay for characterization of dense granule functionality of platelets
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关键字: 疟疾平 ; 盐酸米帕林二盐酸奎吖因 ; 6-氯-9-(4-二乙氨基-1-甲基丁氨基)-2-甲氧基吖啶 二盐酸盐 ; 米帕林 二盐酸盐
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