Product Description
(S)-2-[(S)-2-Amino-2-(tetrahydrofuran-3-yl)acetamido]-2-(tetrahydrofuran-3-yl)acetic Acid is a highly functionalized chiral amino acid building block designed for peptide chemistry and medicinal chemistry applications.
Featuring two stereochemically defined tetrahydrofuran-containing amino acid units, this compound provides a rigid three-dimensional scaffold that can enhance conformational control, improve molecular recognition, and expand chemical diversity during lead optimization. Its multiple functional groups make it suitable for peptide elongation, analogue synthesis, and structure–activity relationship (SAR) studies.
This building block is particularly valuable for the development of peptide therapeutics, macrocycles, enzyme inhibitors, and other biologically active small molecules.
Key Features
Chiral amino acid building block
Dual tetrahydrofuran (THF) motifs
Conformationally constrained scaffold
Suitable for peptide synthesis and medicinal chemistry
Ideal for SAR studies and analogue library construction
Available for custom synthesis and scale-up
中文产品描述
(S)-2-[(S)-2-氨基-2-(四氢呋喃-3-基)乙酰氨基]-2-(四氢呋喃-3-基)乙酸 是一种具有多个手性中心的高级氨基酸砌块,适用于多肽化学、药物化学及创新药研发。
该化合物含有两个 四氢呋喃(THF) 手性单元,可提供刚性的三维空间构象,有助于提高分子识别能力,并丰富先导化合物的结构多样性。其兼具氨基和羧基等活性官能团,可广泛用于多肽延伸、类似物合成以及构效关系(SAR)研究。
Applications
关键字: Amino acid;Chiral;Pharmaceutical inter;Custom synthesis;
**重庆速研医药科技有限公司(Chongqing Rapidsyn Pharmaceutical Technology Co., Ltd.)** 是一家专注于医药化学研发和定制合成服务的高新技术企业。公司拥有经验丰富的研发团队,可提供从毫克(mg)到公斤(kg)级别的定制合成、工艺开发、药物中间体及科研化学品开发服务。
依托专业的技术能力、严格的质量控制和高效的项目管理,重庆速研致力于为全球制药企业、生物技术公司、高校及科研机构提供可靠、高效的化学研发解决方案,帮助客户加速研发进程。