蟾毒灵 MSDS3-b,14-Dihydroxy-5-beta-bufa-20,22-dienolide
Bufalin (0, 1, 2, 4 μM for 48 hours) decreases cell viability in NCI-H460 cells. Bufalin (2 μM) increases caspae-3, Endo G and GADD153 mRNA expression, but decreases the GRP78 mRNA expression.
Cell Viability Assay
Bufalin (0.1, 0.2, or 0.4 mg/kg, i.p., daily for 14 days) shows significant anti-tumor activity in mice bearing NCI-H460 cells.